SCHEMBL1849302

SCHEMBL1849302

O=C(O)Nc1ccc(-c2ccc3scnc3c2)nc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.46
HSD11B1 P28845 1/20 0.46
AURKA O14965 1/20 0.46
PTPN1 P18031 4/20 0.45
PTPN2 P17706 2/20 0.45
RIPK2 O43353 1/20 0.44
EGFR P00533 1/20 0.44
KDR P35968 1/20 0.44
TGFBR1 P36897 1/20 0.44
MCL1 Q07820 5/20 0.43
WNT3A P56704 1/20 0.42
PIK3CD O00329 1/20 0.42
PTPN6 P29350 1/20 0.41
PTPN11 Q06124 1/20 0.41
KEAP1 Q14145 1/20 0.41
NFE2L2 Q16236 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
FFAR1 O14842 1/20 0.41
HIF1A Q16665 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1846865 0.85 RIPK2 (0.54) NAMPTHSD11B1AURKARIPK2EGFR
SCHEMBL3311143 0.83 DYRK2 (0.45) NAMPTHSD11B1AURKAPTPN1RIPK2
SCHEMBL22341666 0.82 HSD11B1 (0.63) NAMPTHSD11B1AURKARIPK2EGFR
SCHEMBL3301474 0.81 RIPK2 (0.43) HSD11B1AURKARIPK2EGFRKDR
SCHEMBL1849737 0.79 AURKA (0.56) NAMPTHSD11B1AURKARIPK2EGFR
SCHEMBL1851318 0.76 TRPV3 (0.44) RIPK2EGFRKDRTGFBR1PIK3CD
SCHEMBL13539289 0.74 NPC1 (0.48) RIPK2KDRTGFBR1PIK3CDNPC1
SCHEMBL13394460 0.74 DYRK1A (0.42) RIPK2EGFRKDRTGFBR1PIK3CD
SCHEMBL22341606 0.73 NPC1 (0.58) NAMPTHSD11B1NPC1RAB9A
SCHEMBL4870704 0.73 PTPN1 (0.67) PTPN1PTPN2WNT3APTPN6PTPN11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2323697-A2 IMAGING AGENTS USEFUL FOR IDENTIFYING AD PATHOLOGY Siemens Medical Solutions USA, Inc. (US) 2011-05-25 EP disclosed
WO-2010011964-A2 IMAGING AGENTS USEFUL FOR IDENTIFYING AD PATHOLOGY SIEMENS MEDICAL SOLUTIONS USA, INC. (US) 2010-01-28 WO disclosed