SCHEMBL1849685

SCHEMBL1849685

CC(C)C(C=O)N(N)c1ncc(C(N)=O)c(Nc2cccc(Br)c2)n1

nearest known ligand 0.59

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SYK P43405 17/20 0.59
CAMK1D Q8IU85 2/20 0.46
AURKA O14965 1/20 0.45
RPS6KB1 P23443 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1354628 1.00 SYK (0.59) SYKCAMK1DAURKARPS6KB1
SCHEMBL1849688 0.90 SYK (0.58) SYKCAMK1DAURKARPS6KB1
SCHEMBL1852547 0.87 SYK (0.60) SYKCAMK1D
SCHEMBL1352375 0.87 SYK (0.61) SYK
SCHEMBL1355333 0.87 SYK (0.60) SYKCAMK1D
SCHEMBL1853033 0.87 SYK (0.61) SYK
SCHEMBL1353406 0.86 SYK (0.61) SYKCAMK1D
SCHEMBL1354029 0.86 SYK (0.64) SYKCAMK1D
SCHEMBL1851695 0.86 SYK (0.61) SYKCAMK1D
SCHEMBL1847521 0.85 SYK (0.62) SYKCAMK1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2323993-A2 2,6-DIAMINO- PYRIMIDIN- 5-YL-CARBOXAMIDES AS SYK OR JAK KINASES INHIBITORS Portola Pharmaceuticals, Inc. (US) 2011-05-25 EP disclosed
WO-2009136995-A2 INHIBITORS OF SYK PROTEIN KINASE PORTOLA PHARMACEUTICALS, INC. (US) 2009-11-12 WO disclosed