SCHEMBL1850820

SCHEMBL1850820

O=C(O)c1ccnc(-c2cccc3cc(COc4cccc(C(F)(F)F)c4)sc23)c1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 2/20 0.54
NR4A2 P43354 2/20 0.52
PPARG P37231 2/20 0.46
KDM4C Q9H3R0 1/20 0.45
MCL1 Q07820 1/20 0.44
S1PR4 O95977 1/20 0.42
S1PR5 Q9H228 1/20 0.42
GPR52 Q9Y2T5 4/20 0.42
ENPP2 Q13822 1/20 0.42
MAOB P27338 1/20 0.41
KMO O15229 1/20 0.41
GPBAR1 Q8TDU6 1/20 0.40
CYSLTR1 Q9Y271 1/20 0.40
LMNA P02545 1/20 0.40
PKM P14618 1/20 0.40
HSD17B10 Q99714 1/20 0.40
AURKA O14965 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1856086 0.89 MEN1 (0.42) MRGPRX4NR4A2GPR52MAOB
SCHEMBL1850062 0.88 MRGPRX4 (0.57) MRGPRX4NR4A2PPARGMCL1S1PR4
SCHEMBL1851849 0.86 GPR52 (0.59) MRGPRX4NR4A2S1PR4S1PR5GPR52
SCHEMBL3219557 0.86 GPR52 (0.61) MRGPRX4GPR52
SCHEMBL1852635 0.85 GPR52 (0.57) MRGPRX4NR4A2KDM4CS1PR4S1PR5
SCHEMBL1850131 0.81 MRGPRX4 (0.49) MRGPRX4NR4A2PPARGMCL1S1PR4
SCHEMBL1849882 0.81 GPR52 (0.57) NR4A2KDM4CS1PR4S1PR5GPR52
SCHEMBL1851239 0.81 GPR52 (0.57) NR4A2KDM4CGPR52
SCHEMBL1850678 0.79 GPR52 (0.56) MRGPRX4NR4A2MCL1S1PR4S1PR5
SCHEMBL1850224 0.79 KDM4C (0.48) KDM4CS1PR4S1PR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2323978-A1 AMIDE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2011-05-25 EP disclosed
WO-2010018874-A1 AMIDE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-02-18 WO disclosed