SCHEMBL1851979

SCHEMBL1851979

CCOC(=O)c1cccc(-c2ccc(F)c3cc(Cc4cc(F)cc(Cl)c4)sc23)c1.O=C(O)c1cccc(-c2ccc(F)c3cc(Cc4cc(F)cc(Cl)c4)sc23)c1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GPR52 Q9Y2T5 3/20 0.53
NPC1 O15118 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TP53 P04637 2/20 0.36
POLB P06746 1/20 0.36
HPGD P15428 1/20 0.36
PTGER1 P34995 1/20 0.36
ALOX5 P09917 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
AKR1C3 P42330 1/20 0.35
AKR1C2 P52895 1/20 0.35
GALR1 P47211 1/20 0.35
EIF4EBP1 Q13541 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1847924 0.97 GPR52 (0.56) GPR52NPC1ALDH1A1MAPTRAB9A
SCHEMBL1867001 0.94 GPR52 (0.53) GPR52NPC1ALDH1A1MAPTRAB9A
SCHEMBL1849783 0.91 GPR52 (0.56) GPR52PTGER1AKR1C3AKR1C2EIF4EBP1
SCHEMBL1851960 0.91 GPR52 (0.55) GPR52NPC1ALDH1A1MAPTRAB9A
SCHEMBL1856025 0.90 GPR52 (0.41) GPR52NPC1ALDH1A1MAPTRAB9A
SCHEMBL1849690 0.89 GPR52 (0.49) GPR52NPC1ALDH1A1MAPTRAB9A
SCHEMBL1851933 0.87 GPR52 (0.53) GPR52NPC1RAB9APTGER1AKR1C3
SCHEMBL1850522 0.86 GPR52 (0.70) GPR52NPC1ALDH1A1MAPTRAB9A
SCHEMBL1848327 0.86 GPR52 (0.44) GPR52NPC1ALDH1A1MAPTRAB9A
SCHEMBL1859640 0.85 GPR52 (0.47) GPR52NPC1ALDH1A1MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2323978-A1 AMIDE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2011-05-25 EP disclosed
WO-2010018874-A1 AMIDE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-02-18 WO disclosed