SCHEMBL18520105

SCHEMBL18520105

Nc1ccc(-c2cnn(C(F)F)c2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
TP53 P04637 2/20 0.41
CYP3A4 P08684 2/20 0.41
TDP1 Q9NUW8 2/20 0.41
CREBBP Q92793 4/20 0.39
BRD4 O60885 2/20 0.39
PIK3CD O00329 2/20 0.38
PIK3CA P42336 2/20 0.38
PIK3CG P48736 2/20 0.38
PIP5K1C O60331 1/20 0.38
PI4KA P42356 1/20 0.38
PI4KB Q9UBF8 1/20 0.38
HSD17B10 Q99714 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
NPC1 O15118 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
RAB9A P51151 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17806585 0.82 CREBBP (0.40) TP53CREBBPBRD4PIK3CDPIK3CA
SCHEMBL17809810 0.81 CREBBP (0.39) ALDH1A1CREBBPBRD4PIK3CDPIK3CA
SCHEMBL22165237 0.81 PIK3CD (0.55) ALDH1A1TP53CYP3A4TDP1CREBBP
SCHEMBL28511565 0.81 PIK3CD (0.44) ALDH1A1PIK3CDPIK3CAPIK3CGPIP5K1C
SCHEMBL30640940 0.81 PIK3CD (0.44) ALDH1A1PIK3CDPIK3CAPIK3CGPIP5K1C
SCHEMBL18520131 0.80 ALOX5AP (0.44) CREBBPBRD4PIK3CDPIK3CAPIK3CG
SCHEMBL20456818 0.77 DRD1 (0.45) ALDH1A1CREBBPBRD4KDM4ESMN1; SMN2
SCHEMBL30888279 0.77 ALDH1A1 (0.52) ALDH1A1CYP3A4TDP1BRD4PIK3CD
SCHEMBL23535770 0.76 BCL2L1 (0.46) TP53CREBBPBRD4HSD17B10KDM4E
SCHEMBL30695445 0.74 DYRK1A (0.45) PIK3CDPIK3CAPIK3CGPIP5K1CPI4KA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017024996-A1 HYDROXY AMIDINE DERIVATIVE, PREPARATION METHOD AND USE IN MEDICINE THEREOF 江苏恒瑞医药股份有限公司 2017-02-16 WO disclosed