SCHEMBL18520752

SCHEMBL18520752

Cc1cc2nccc(OS(=O)(=O)C(F)(F)F)c2c(C)c1Br

nearest known ligand 0.37

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.37
SLC22A12 Q96S37 1/20 0.33
SCN9A Q15858 1/20 0.31
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
EPAS1 Q99814 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14999154 0.78 SRC (0.39) ESR2SLC22A12SCN9A
SCHEMBL18498954 0.75 NQO2 (0.37) ESR2
SCHEMBL18520603 0.73 ALDH1A1 (0.44) ESR2
SCHEMBL29069658 0.72 SLC22A12 (0.34) ESR2SLC22A12CA1CA2
SCHEMBL12367211 0.71 HTR1A (0.41) ESR2SLC22A12CA1CA2
SCHEMBL4490029 0.71 SLC22A12 (0.47) ESR2SLC22A12CA1CA2
SCHEMBL3851998 0.71 SLC22A12 (0.56) ESR2SLC22A12CA1CA2
SCHEMBL244619 0.70 PDGFRB (0.48) CA1CA2
SCHEMBL244158 0.70 ALDH1A1 (0.36) SLC22A12CA1CA2
SCHEMBL15125302 0.70 PDE4A (0.35) ESR2CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017027768-A1 COMPOSITIONS AND METHODS FOR TREATING TUBERCULOSIS THE BROAD INSTITUTE, INC. (US) 2017-02-16 WO disclosed