SCHEMBL1853064

SCHEMBL1853064

Cc1c(Cc2cccc(C(F)(F)F)c2)sc2c(-c3cc(C(=O)O)ccn3)cccc12.Cc1c(Cc2cccc(C(F)(F)F)c2)sc2c(-c3cc(C(N)=O)ccn3)cccc12

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 1/20 0.48
GPR52 Q9Y2T5 10/20 0.47
NR4A2 P43354 1/20 0.41
ROCK1 Q13464 2/20 0.41
AURKA O14965 1/20 0.40
RPS6KB1 P23443 1/20 0.40
AURKB Q96GD4 1/20 0.40
NR3C2 P08235 1/20 0.39
MRGPRX4 Q96LA9 1/20 0.39
MAOB P27338 1/20 0.39
LIPG Q9Y5X9 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3217369 0.97 GPR52 (0.50) KDM4CGPR52ROCK1AURKARPS6KB1
SCHEMBL1856110 0.97 KDM4C (0.51) KDM4CGPR52NR4A2ROCK1MRGPRX4
SCHEMBL1850776 0.91 KDM4C (0.46) KDM4CGPR52NR4A2ROCK1MRGPRX4
SCHEMBL1849782 0.88 KDM4C (0.43) KDM4CGPR52NR4A2ROCK1MRGPRX4
SCHEMBL3209831 0.87 ROCK1 (0.43) KDM4CGPR52ROCK1MRGPRX4
SCHEMBL1856629 0.84 GPR52 (0.56) GPR52
SCHEMBL1850602 0.84 GPR52 (0.49) GPR52NR4A2MRGPRX4LIPG
SCHEMBL1852235 0.84 GPR52 (0.54) GPR52MAOB
SCHEMBL1849882 0.83 GPR52 (0.57) KDM4CGPR52NR4A2
SCHEMBL1852456 0.80 GPR52 (0.46) GPR52MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2323978-A1 AMIDE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2011-05-25 EP disclosed
WO-2010018874-A1 AMIDE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-02-18 WO disclosed