SCHEMBL185404

SCHEMBL185404

CC(=O)NC(c1ccccc1C)C(C)C

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.44
ALOX12 P18054 1/20 0.44
RAB9A P51151 1/20 0.44
NCOA3 Q9Y6Q9 1/20 0.44
ALDH1A1 P00352 2/20 0.43
HPGD P15428 1/20 0.43
MTNR1A P48039 6/20 0.39
MTNR1B P49286 6/20 0.39
ESR1 P03372 1/20 0.38
CYP1A2 P05177 1/20 0.38
ACP3 P15309 1/20 0.38
CTSA P10619 1/20 0.37
NR3C2 P08235 1/20 0.37
HDAC1 Q13547 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7723692 0.81 ALDH1A1 (0.46) ALDH1A1HPGDMTNR1AMTNR1B
SCHEMBL185646 0.76 HDAC1 (0.60) ALDH1A1HPGDMTNR1AMTNR1BHDAC1
SCHEMBL16371412 0.75 ALDH1A1 (0.43) ALDH1A1HPGDMTNR1AMTNR1BESR1
SCHEMBL25509348 0.75 ESR1 (0.45) ALDH1A1ESR1ACP3NR3C2
SCHEMBL185423 0.74 CTSA (0.44) ALDH1A1HPGDCTSA
SCHEMBL15116640 0.72 ESR1 (0.42) NPC1RAB9AALDH1A1HPGDESR1
SCHEMBL11294913 0.72 ALDH1A1 (0.46) ALDH1A1ESR1ACP3CTSAHDAC1
SCHEMBL185644 0.71 CTSA (0.42) ALDH1A1CTSA
SCHEMBL15695548 0.71 ESR1 (0.45) NPC1RAB9AALDH1A1HPGDESR1
Hydrochloric Acid SCHEMBL4329941 0.70 ALDH1A1 (0.45) ALDH1A1ESR1ACP3CTSAHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401260-A1 DIOXO-IMIDAZOLIDINE DERIVATIVES, WHICH INHIBIT THE ENZYME SOAT-1, AND PHARMACEUTICAL AND COSMETIC COMPOSITIONS CONTAINING THEM Galderma Research & Development (FR) 2012-01-04 EP claimed
WO-2010097465-A1 DIOXO-IMIDAZOLIDINE DERIVATIVES, WHICH INHIBIT THE ENZYME SOAT-1, AND PHARMACEUTICAL AND COSMETIC COMPOSITIONS CONTAINING THEM GALDERMA RESEARCH & DEVELOPMENT (FR) 2010-09-02 WO claimed
EP-2401260-A1 DIOXO-IMIDAZOLIDINE DERIVATIVES, WHICH INHIBIT THE ENZYME SOAT-1, AND PHARMACEUTICAL AND COSMETIC COMPOSITIONS CONTAINING THEM Galderma Research & Development (FR) 2012-01-04 EP disclosed
WO-2010097465-A1 DIOXO-IMIDAZOLIDINE DERIVATIVES, WHICH INHIBIT THE ENZYME SOAT-1, AND PHARMACEUTICAL AND COSMETIC COMPOSITIONS CONTAINING THEM GALDERMA RESEARCH & DEVELOPMENT (FR) 2010-09-02 WO disclosed