SCHEMBL1854343

SCHEMBL1854343

O=C(CCCCBr)Nc1cc(-c2cccc(Br)c2)n[nH]1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 15/20 0.49
HDAC2 Q92769 12/20 0.49
HDAC8 Q9BY41 10/20 0.47
HDAC6 Q9UBN7 8/20 0.47
HDAC3 O15379 7/20 0.47
HDAC10 Q969S8 6/20 0.47
HDAC4 P56524 3/20 0.47
HDAC7 Q8WUI4 3/20 0.47
HDAC11 Q96DB2 3/20 0.47
HDAC9 Q9UKV0 3/20 0.47
HDAC5 Q9UQL6 3/20 0.47
MEN1 O00255 1/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
HTT P42858 1/20 0.41
KMT2A Q03164 1/20 0.41
IDO1 P14902 1/20 0.40
METAP2 P50579 1/20 0.40
NPC1 O15118 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1859648 0.83 CHRNA3 (0.57)
SCHEMBL16150892 0.80 MEN1 (0.48) MEN1LMNAMAPTHPGDHTT
SCHEMBL1852946 0.78 HDAC1 (0.53) HDAC1HDAC2HDAC8HDAC6HDAC3
SCHEMBL2055601 0.78 KCNH2 (0.53)
SCHEMBL16151050 0.73 MAPT (0.42) HDAC1HDAC2HDAC8HDAC3HDAC10
SCHEMBL21805191 0.73 GAA (0.62) HDAC1HDAC2HDAC8HDAC6HDAC3
SCHEMBL30087930 0.73 GAA (0.62) HDAC1HDAC2HDAC8HDAC6HDAC3
SCHEMBL14922960 0.72 HDAC1 (0.44) HDAC1HDAC2HDAC8HDAC6HDAC3
SCHEMBL2055612 0.71 ALDH1A1 (0.52)
SCHEMBL2055616 0.71 ALDH1A1 (0.52)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8163729-B2 Modulators of α7 nicotinic acetylcholine receptors and therapeutic uses thereof WYETH (US) 2012-04-24 US disclosed
EP-2323988-A1 ALPHA7 NICOTINIC ACETYLCHOLINE RECEPTOR INHIBITORS Wyeth LLC (US) 2011-05-25 EP disclosed