SCHEMBL18544256

SCHEMBL18544256

O=c1cnc2ccc(F)cc2n1I

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.38
ALDH1A1 P00352 2/20 0.36
USP2 O75604 1/20 0.36
LMNA P02545 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
TSHR P16473 1/20 0.36
CYP2C19 P33261 1/20 0.36
GRIN2B Q13224 8/20 0.36
BRD4 O60885 1/20 0.36
GRIN1 Q05586 1/20 0.35
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35
DAO P14920 1/20 0.34
KDM4E B2RXH2 1/20 0.34
HPGD P15428 1/20 0.34
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19231294 0.81 CYP11B1 (0.44) PARP1ALDH1A1USP2CYP1A2CYP3A4
SCHEMBL29489040 0.77 CYP11B1 (0.48) ALDH1A1USP2LMNACYP1A2CYP3A4
SCHEMBL14313795 0.77 CYP11B1 (0.48) ALDH1A1USP2LMNACYP1A2CYP3A4
SCHEMBL21202580 0.77 GRIN2B (0.37) PARP1ALDH1A1USP2LMNACYP1A2
SCHEMBL2799084 0.74 ALDH1A1 (0.40) ALDH1A1USP2LMNACYP1A2CYP3A4
SCHEMBL3859045 0.73 ALDH1A1 (0.39) ALDH1A1USP2LMNACYP1A2CYP3A4
SCHEMBL15850934 0.72 ALDH1A1 (0.39) ALDH1A1USP2LMNACYP1A2CYP3A4
SCHEMBL19706890 0.72 OPRM1 (0.48) ALDH1A1KDM4ECYP11B1CYP11B2
SCHEMBL19212760 0.71 GRIN2B (0.47) ALDH1A1USP2LMNACYP1A2CYP3A4
SCHEMBL18544279 0.71 HPGD (0.42) ALDH1A1LMNATSHRPDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017029602-A2 COMPOUNDS FOR USE IN ANTIBACTERIAL APPLICATIONS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2017-02-23 WO disclosed