SCHEMBL18544288

SCHEMBL18544288

COc1cc(F)c2nccc(I)c2c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.38
CCR5 P51681 1/20 0.38
CCR8 P51685 1/20 0.38
ACVR1 Q04771 1/20 0.37
PDE10A Q9Y233 4/20 0.37
PDE2A O00408 3/20 0.37
KDM4E B2RXH2 2/20 0.36
NOS3 P29474 1/20 0.36
NOS1 P29475 1/20 0.36
NOS2 P35228 1/20 0.36
TRPA1 O75762 1/20 0.35
TAAR1 Q96RJ0 1/20 0.35
CYP1A1 P04798 2/20 0.35
CYP1A2 P05177 2/20 0.35
CYP1B1 Q16678 2/20 0.35
CYP2E1 P05181 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C8 P10632 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2A6 P11509 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29923344 0.82 CCR1 (0.39) CCR1CCR5CCR8KDM4ENOS3
SCHEMBL3375901 0.81 CCR1 (0.38) CCR1CCR5CCR8ACVR1PDE10A
SCHEMBL2923376 0.81 NOS3 (0.40) CCR1CCR5CCR8ACVR1PDE10A
SCHEMBL4279169 0.81 NOS3 (0.43) CCR1CCR5CCR8ACVR1PDE10A
Hydrochloric Acid SCHEMBL5748572 0.79 NOS3 (0.42) CCR1CCR5CCR8ACVR1PDE10A
Hydrochloric Acid SCHEMBL6640376 0.79 NOS3 (0.42) CCR1CCR5CCR8ACVR1PDE10A
SCHEMBL20687484 0.78 CA1 (0.39) CCR1CCR5CCR8ACVR1PDE10A
SCHEMBL27588449 0.78 KDM4E (0.60) KDM4ELMNA
SCHEMBL20277757 0.78 CDK8 (0.43) PDE10AKDM4ETRPA1CYP1A2CYP3A4
SCHEMBL3375976 0.77 CCR1 (0.49) CCR1CCR5CCR8ACVR1PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017029602-A2 COMPOUNDS FOR USE IN ANTIBACTERIAL APPLICATIONS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2017-02-23 WO disclosed