SCHEMBL29923344

SCHEMBL29923344

COc1cc(Br)c2nccc(I)c2c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.39
CCR5 P51681 1/20 0.39
CCR8 P51685 1/20 0.39
KDM4E B2RXH2 5/20 0.37
NOS3 P29474 1/20 0.37
NOS1 P29475 1/20 0.37
NOS2 P35228 1/20 0.37
CYP1A1 P04798 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2E1 P05181 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C8 P10632 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2A6 P11509 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP4B1 P13584 1/20 0.36
CYP2B6 P20813 1/20 0.36
CYP3A5 P20815 1/20 0.36
CYP2A7 P20853 1/20 0.36
CYP3A7 P24462 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18544288 0.82 CCR1 (0.38) CCR1CCR5CCR8KDM4ENOS3
SCHEMBL24916289 0.81 NSD2 (0.50) CCR1CCR5CCR8KDM4ENOS3
SCHEMBL29924149 0.80 NOS3 (0.41) CCR1CCR5CCR8KDM4ENOS3
SCHEMBL24916103 0.80 NOS3 (0.41) CCR1CCR5CCR8KDM4ENOS3
SCHEMBL29923920 0.80 HSP90AA1 (0.50) CCR1CCR5CCR8KDM4ENOS3
SCHEMBL5262975 0.73 PDGFRB (0.42) CCR1CCR5CCR8KDM4ENOS3
SCHEMBL17502532 0.73 NSD2 (0.40) CCR1CCR5CCR8NOS3NOS1
SCHEMBL29923869 0.73 PDGFRB (0.42) CCR1CCR5CCR8KDM4ENOS3
SCHEMBL24916137 0.73 NSD2 (0.38) CCR1CCR5CCR8KDM4ENOS3
SCHEMBL29923321 0.73 NSD2 (0.38) CCR1CCR5CCR8KDM4ENOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4055013-A1 WDR5 INHIBITORS AND MODULATORS Vanderbilt University (US) 2022-09-14 EP disclosed