SCHEMBL1854946

SCHEMBL1854946

CS(=O)(=O)NCc1c[nH]c2ccccc12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MC1R Q01726 3/20 0.54
MC5R P33032 2/20 0.54
MC3R P41968 1/20 0.54
GPR84 Q9NQS5 3/20 0.54
CYP19A1 P11511 2/20 0.54
MEN1 O00255 4/20 0.53
KMT2A Q03164 4/20 0.53
MAPT P10636 2/20 0.53
CYP3A4 P08684 2/20 0.53
AHR P35869 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
KDM4E B2RXH2 3/20 0.51
ALDH1A1 P00352 2/20 0.51
HTR1A P08908 1/20 0.51
HTR2A P28223 1/20 0.51
HTT P42858 1/20 0.51
IDO1 P14902 1/20 0.51
CYP2D6 P10635 1/20 0.50
TSHR P16473 1/20 0.50
CYP2C19 P33261 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL760892 0.84 CYP19A1 (0.70) MC1RMC5RMC3RCYP19A1MEN1
SCHEMBL19410682 0.82 ALOX12 (0.62) CYP19A1MEN1KMT2AKDM4EALDH1A1
SCHEMBL25252806 0.81 CYP19A1 (0.74) MC1RMC5RMC3RCYP19A1
SCHEMBL25241467 0.80 CYP19A1 (0.50) MC1RMC5RMC3RCYP19A1
SCHEMBL25247387 0.80 NR3C1 (0.66) CYP19A1MEN1KMT2AMAPTCYP3A4
SCHEMBL1851985 0.78 KMT2A (0.58) GPR84CYP19A1MEN1KMT2AMAPT
SCHEMBL29350522 0.78 HTR2A (0.69) MC1RMC5RMC3RGPR84MEN1
SCHEMBL1092334 0.78 HTR2A (0.69) MC1RMC5RMC3RGPR84MEN1
SCHEMBL25247095 0.77 MGAM (0.52) MC1RMC5RMC3RGPR84CYP19A1
SCHEMBL25244099 0.77 CYP19A1 (0.60) CYP19A1MEN1KMT2AMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250093329-A1 SCREENING OF COMPOUNDS THE UNIVERSITY OF TULSA 2025-03-20 US disclosed
US-20230266302-A1 SYNTHESIS AND USE OF N-BENZYL SULFONAMIDES THE UNIV OF TULSA (US) 2023-08-24 US disclosed
EP-4185706-A1 SYNTHESIS AND USE OF N-BENZYL SULFONAMIDES The University Of Tulsa (US) 2023-05-31 EP disclosed
US-8242116-B2 Fused thiazole derivatives as kinase inhibitors UCB PHARMA S.A. (BE) 2012-08-14 US disclosed
EP-2035436-B1 FUSED THIAZOLE DERIVATIVES AS KINASE INHIBITORS UCB PHARMA SA (BE) 2011-05-25 EP disclosed
US-20100137302-A1 Fused Thiazole Derivatives as Kinase Inhibitors UCB PHARMA S.A. (BE) 2010-06-03 US disclosed
WO-2009122148-A1 FUSED THIOPHENE AND THIAZOLE DERIVATIVES AS PI3K KINASE INHIBITORS UCB PHARMA S.A. (BE) 2009-10-08 WO disclosed
WO-2009071895-A1 FUSED THIAZOLE AND THIOPHENE DERIVATIVES AS KINASE INHIBITORS UCB PHARMA S.A. (BE) 2009-06-11 WO disclosed
WO-2009071890-A1 TRICYCLIC KINASE INHIBITORS UCB PHARMA S.A. (BE) 2009-06-11 WO disclosed
WO-2009071888-A1 PYRROLOTHIAZOLES AS PI3-KINASE INHIBITORS UCB PHARMA S.A. (BE) 2009-06-11 WO disclosed
EP-2035436-A1 FUSED THIAZOLE DERIVATIVES AS KINASE INHIBITORS UCB Pharma S.A. (BE) 2009-03-18 EP disclosed
WO-2008001076-A1 FUSED THIAZOLE DERIVATIVES AS KINASE INHIBITORS UCB PHARMA S.A. (BE) 2008-01-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100137302-A1 Fused Thiazole Derivatives as Kinase Inhibitors PI4KA, PDPK1, PIK3CA MC1R 1148/4885MC5R 1446/4885MC3R 1154/4885
US-20230266302-A1 SYNTHESIS AND USE OF N-BENZYL SULFONAMIDES ATP5ME, ATP5F1B, ATP5MG MC1R 4670/4885MC5R 4786/4885MC3R 4854/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.