SCHEMBL1855101

SCHEMBL1855101

COc1ccc(-c2cc(N)n(C(=O)O)n2)cn1

nearest known ligand 0.67

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KLK3 P07288 8/20 0.67
F2 P00734 1/20 0.60
MKNK1 Q9BUB5 1/20 0.49
MKNK2 Q9HBH9 1/20 0.49
PIK3CA P42336 6/20 0.45
MTOR P42345 1/20 0.44
KCNH2 Q12809 2/20 0.43
JAK2 O60674 1/20 0.43
NNMT P40261 1/20 0.43
HSD17B1 P14061 1/20 0.42
HSD17B2 P37059 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1853581 0.84 KLK3 (0.61) KLK3F2MKNK1MKNK2PIK3CA
SCHEMBL25409385 0.81 KLK3 (0.57) KLK3F2MKNK1MKNK2PIK3CA
SCHEMBL26847558 0.70 KLK3 (0.45) KLK3F2MKNK1MKNK2PIK3CA
SCHEMBL3754419 0.68 CYP2A6 (0.68) MKNK1MKNK2PIK3CANNMTHSD17B1
SCHEMBL31174412 0.68 CYP2A6 (0.68) MKNK1MKNK2PIK3CANNMTHSD17B1
SCHEMBL2469483 0.68 MKNK1 (0.46) KLK3MKNK1MKNK2PIK3CAMTOR
SCHEMBL1852996 0.68 KLK3 (0.44) KLK3F2PIK3CA
SCHEMBL24029943 0.68 MKNK1 (0.49) KLK3MKNK1MKNK2PIK3CAMTOR
SCHEMBL16835945 0.67 MKNK1 (0.51) KLK3MKNK1MKNK2PIK3CAKCNH2
SCHEMBL29365356 0.67 MKNK1 (0.73) MKNK1MKNK2NNMTHSD17B1HSD17B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2323988-A1 ALPHA7 NICOTINIC ACETYLCHOLINE RECEPTOR INHIBITORS Wyeth LLC (US) 2011-05-25 EP disclosed
WO-2010009290-A1 ALPHA7 NICOTINIC ACETYLCHOLINE RECEPTOR INHIBITORS WYETH (US) 2010-01-21 WO disclosed