SCHEMBL1855458

SCHEMBL1855458

CC(N)C(O)O.O=C(NC(CO)CO)c1cccc(-c2cccc3cc(Cc4cccc(C(F)(F)F)c4)oc23)c1

nearest known ligand 0.69

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GPR52 Q9Y2T5 13/20 0.69
TAS1R3 Q7RTX0 1/20 0.41
TAS1R1 Q7RTX1 1/20 0.41
PIN1 Q13526 1/20 0.41
NPSR1 Q6W5P4 1/20 0.40
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
CYP1A2 P05177 1/20 0.37
CYP2C19 P33261 1/20 0.37
ALDH1A1 P00352 1/20 0.37
CTSL P07711 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3209952 0.94 GPR52 (0.76) GPR52TAS1R3TAS1R1PIN1NPSR1
SCHEMBL1851771 0.81 GPR52 (1.00) GPR52
SCHEMBL1849964 0.80 GPR52 (0.75) GPR52ALDH1A1
SCHEMBL3206803 0.79 GPR52 (0.81) GPR52ALDH1A1
SCHEMBL1856609 0.77 GPR52 (0.79) GPR52ALDH1A1
SCHEMBL3209943 0.77 GPR52 (0.79) GPR52ALDH1A1
SCHEMBL1846506 0.77 GPR52 (0.81) GPR52ALDH1A1
SCHEMBL1852519 0.75 GPR52 (0.68) GPR52ALDH1A1
SCHEMBL3213465 0.74 GPR52 (0.62) GPR52CYP1A2CYP2C19
SCHEMBL1848289 0.72 GPR52 (0.81) GPR52

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2323978-A1 AMIDE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2011-05-25 EP disclosed
WO-2010018874-A1 AMIDE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-02-18 WO disclosed