SCHEMBL185548

SCHEMBL185548

NC1(OC(=O)NCc2ccc(Nc3ccccc3C(F)(F)F)cc2)COC1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
HTT P42858 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
GAA P10253 2/20 0.38
POLB P06746 4/20 0.37
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
KDM4E B2RXH2 3/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
THRB P10828 1/20 0.36
NOX1 Q9Y5S8 1/20 0.36
LMNA P02545 2/20 0.36
NAMPT P43490 2/20 0.36
MT-CO2 P00403 1/20 0.36
TSHR P16473 1/20 0.35
AURKA O14965 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2805090 0.85 ALDH1A1 (0.43) ALDH1A1MAPTHPGDHTTNPSR1
SCHEMBL185458 0.82 ALDH1A1 (0.39) ALDH1A1MAPTHPGDHTTNPSR1
SCHEMBL184945 0.80 MT-CO2 (0.43) ALDH1A1MAPTHPGDHTTNPSR1
SCHEMBL185024 0.80 OPRL1 (0.36) GAAPOLBRAB9AKMT2AAURKA
SCHEMBL2805680 0.79 ALDH1A1 (0.40) ALDH1A1MAPTHPGDHTTNPSR1
SCHEMBL186501 0.79 ALDH1A1 (0.40) ALDH1A1MAPTHPGDHTTNPSR1
SCHEMBL186385 0.79 CYP1A2 (0.38) MAPTGAAPOLBRAB9AKDM4E
SCHEMBL185956 0.78 SIRT2 (0.36) ALDH1A1GAARAB9AKMT2ALMNA
SCHEMBL2781755 0.76 POLB (0.40) ALDH1A1MAPTHPGDHTTNPSR1
SCHEMBL185629 0.76 POLB (0.36) ALDH1A1HPGDGAAPOLBNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401256-B1 Compounds as bradykinin B1 antagonists BOEHRINGER INGELHEIM INT (DE) 2013-04-17 EP disclosed
EP-2401256-A1 COMPOUNDS AS BRADYKININ B1 ANTAGONISTS Boehringer Ingelheim International GmbH (DE) 2012-01-04 EP disclosed
WO-2010097372-A1 COMPOUNDS AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed