SCHEMBL18558296

SCHEMBL18558296

CNC(O)c1ccc(C#N)cn1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
S1PR3 Q99500 6/20 0.38
LMNA P02545 1/20 0.36
GAA P10253 1/20 0.36
KCNJ1 P48048 5/20 0.35
KCNH2 Q12809 1/20 0.35
LOXL2 Q9Y4K0 1/20 0.35
CYP19A1 P11511 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
S1PR1 P21453 2/20 0.34
PANK3 Q9H999 1/20 0.34
GRIN1 Q05586 1/20 0.34
GRIN2B Q13224 1/20 0.34
S1PR4 O95977 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22481395 0.80 ALDH1A1 (0.43) KDM4EALDH1A1L3MBTL1S1PR3LMNA
SCHEMBL22481391 0.77 KCNJ1 (0.43) KDM4EALDH1A1L3MBTL1S1PR3KCNJ1
SCHEMBL2737290 0.76 ALDH1A1 (0.46) KDM4EALDH1A1L3MBTL1S1PR3LMNA
SCHEMBL18558695 0.74 APLNR (0.50) KCNH2
SCHEMBL18558292 0.73 PTK2 (0.41) L3MBTL1S1PR3S1PR1S1PR4
SCHEMBL22538435 0.73 ALDH1A1 (0.43) KDM4EALDH1A1L3MBTL1S1PR3LMNA
SCHEMBL29872319 0.73 ALDH1A1 (0.43) KDM4EALDH1A1L3MBTL1S1PR3LMNA
SCHEMBL20447635 0.73 ALDH1A1 (0.43) KDM4EALDH1A1L3MBTL1S1PR3LMNA
SCHEMBL15486717 0.73 ALDH1A1 (0.43) KDM4EALDH1A1L3MBTL1S1PR3LMNA
SCHEMBL19574036 0.73 ALDH1A1 (0.43) KDM4EALDH1A1L3MBTL1S1PR3LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9580433-B2 4-amino-6-phenyl-5,6-dihydroimidazo[1,5-A]pyrazine derivatives as inhibitors of beta-secretase (BACE) JANSSEN PHARMACEUTICA NV (BE) 2017-02-28 US disclosed