SCHEMBL185693

SCHEMBL185693

CNc1ncc(OC(=O)N[C@@]2(C(=O)NCc3ncc(Nc4c(F)cccc4C(F)(F)F)cc3Cl)CCOC2)cn1

nearest known ligand 0.33

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
FGFR4 P22455 1/20 0.33
CCNC P24863 1/20 0.33
CDK8 P49336 1/20 0.33
P2RX7 Q99572 1/20 0.32
JAK1 P23458 2/20 0.31
JAK3 P52333 2/20 0.31
JAK2 O60674 1/20 0.31
OPRL1 P41146 2/20 0.31
BTK Q06187 1/20 0.31
TRPV1 Q8NER1 4/20 0.31
FAAH O00519 3/20 0.31
EGFR P00533 1/20 0.30
LRRK2 Q5S007 1/20 0.30
MAP4K1 Q92918 1/20 0.30
PTGES O14684 1/20 0.30
SYK P43405 2/20 0.30
P2RX3 P56373 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14857218 0.92 MAPK7 (0.32) FGFR4P2RX7OPRL1TRPV1FAAH
SCHEMBL2806537 0.90 P2RX7 (0.34) CCNCCDK8P2RX7JAK1JAK3
SCHEMBL14856567 0.89 OPRL1 (0.35) CCNCCDK8OPRL1TRPV1FAAH
SCHEMBL14856773 0.87 CNR2 (0.34) CCNCCDK8P2RX7TRPV1FAAH
SCHEMBL14856726 0.86 FAAH (0.35) FGFR4CCNCCDK8JAK1JAK3
SCHEMBL2807071 0.85 BDKRB1 (0.35) P2RX7OPRL1PTGES
SCHEMBL185684 0.85 BDKRB1 (0.35) P2RX7OPRL1PTGES
Hydrochloric Acid SCHEMBL185917 0.85 FAAH (0.32) OPRL1TRPV1FAAH
SCHEMBL2810139 0.84 BDKRB1 (0.36) P2RX7OPRL1EGFRPTGES
SCHEMBL186187 0.84 TRPV1 (0.36) P2RX7TRPV1FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401256-A1 COMPOUNDS AS BRADYKININ B1 ANTAGONISTS Boehringer Ingelheim International GmbH (DE) 2012-01-04 EP disclosed
WO-2010097372-A1 COMPOUNDS AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed