SCHEMBL18596173

SCHEMBL18596173

C=C(N)C1CCCN(C(=O)C(C)C)C1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.42
MAPK1 P28482 1/20 0.42
LMNA P02545 1/20 0.41
CHRNB2 P17787 1/20 0.39
CHRNA3 P32297 1/20 0.39
CHRNA4 P43681 1/20 0.39
CHRNB3 Q05901 1/20 0.39
CHRNA6 Q15825 1/20 0.39
GLA P06280 1/20 0.38
HSD17B10 Q99714 1/20 0.38
GAA P10253 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
CA12 O43570 3/20 0.36
CA1 P00915 3/20 0.36
CA2 P00918 3/20 0.36
CA9 Q16790 3/20 0.36
ITGB3 P05106 3/20 0.36
ITGA2B P08514 3/20 0.36
PDE4B Q07343 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10311690 0.87 ALDH1A1 (0.55) ALDH1A1MAPK1LMNACHRNB2CHRNA3
SCHEMBL12741548 0.81 CHRNB2 (0.42) ALDH1A1MAPK1LMNACHRNB2CHRNA3
SCHEMBL12430299 0.81 ALDH1A1 (0.46) ALDH1A1MAPK1CHRNB2CHRNA3CHRNA4
SCHEMBL14348127 0.78 ALDH1A1 (0.44) ALDH1A1MAPK1LMNACHRNB2CHRNA3
SCHEMBL25919918 0.77 BCHE (0.47) ALDH1A1CHRNB2CHRNA3CHRNA4CHRNB3
SCHEMBL12788623 0.77 ALDH1A1 (0.42) ALDH1A1MAPK1LMNAGLAHSD17B10
SCHEMBL18610409 0.76 GAA (0.46) ALDH1A1MAPK1LMNACHRNB2CHRNA3
SCHEMBL12413686 0.76 CHRNB2 (0.43) ALDH1A1LMNACHRNB2CHRNA3CHRNA4
SCHEMBL478900 0.76 CHRNB2 (0.43) ALDH1A1MAPK1LMNACHRNB2CHRNA3
SCHEMBL12414281 0.76 CHRNB2 (0.43) ALDH1A1LMNACHRNB2CHRNA3CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9586956-B2 Isoquinoline and naphthyridine derivatives GENENTECH, INC. (US) 2017-03-07 US disclosed