SCHEMBL18600085

SCHEMBL18600085

CC(C)(C)OC(=O)N=CC1CCN(c2ccccc2N)C1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.46
MEN1 O00255 1/20 0.46
USP2 O75604 1/20 0.46
KMT2A Q03164 1/20 0.46
ADRA2C P18825 1/20 0.39
PIM1 P11309 1/20 0.38
PIM3 Q86V86 1/20 0.38
PIM2 Q9P1W9 1/20 0.38
GPR119 Q8TDV5 3/20 0.38
KEAP1 Q14145 1/20 0.38
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 2/20 0.35
NPC1 O15118 1/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35
RAB9A P51151 1/20 0.35
KDM1A O60341 1/20 0.35
NOTUM Q6P988 2/20 0.34
POLB P06746 1/20 0.34
NR4A1 P22736 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18600082 0.83 LMNA (0.50) MEN1KMT2AGPR119ALDH1A1MAPT
SCHEMBL23368546 0.75 GAA (0.55) GAAMEN1USP2KMT2AADRA2C
SCHEMBL3211670 0.74 PIM1 (0.60) GAAMEN1USP2KMT2APIM1
SCHEMBL3211686 0.74 PIM1 (0.60) GAAMEN1USP2KMT2APIM1
SCHEMBL14206408 0.74 PIM1 (0.60) GAAMEN1USP2KMT2APIM1
SCHEMBL6311733 0.73 KEAP1 (0.47) GAAMEN1USP2KMT2AADRA2C
SCHEMBL1271996 0.72 CKS1B (0.55) GAAMEN1USP2KMT2APIM1
SCHEMBL9984095 0.72 PIM1 (0.48) GAAMEN1USP2KMT2AADRA2C
SCHEMBL14207419 0.72 CKS1B (0.52) GAAMEN1USP2KMT2AKDM4E
SCHEMBL23107339 0.72 MAP4K4 (0.36) GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2078003-B1 ANILINOPIPERAZINE DERIVATIVES AND METHODS OF USE THEREOF MERCK SHARP & DOHME (US) 2017-03-08 EP disclosed