SCHEMBL18600237

SCHEMBL18600237

N=C/C=C\Nc1ccccc1NC(=O)c1csc(-c2cccs2)n1

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
CHEK1 O14757 6/20 0.55
KDM4E B2RXH2 4/20 0.51
HDAC3 O15379 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
IRAK4 Q9NWZ3 4/20 0.43
NPC1 O15118 3/20 0.42
TDP1 Q9NUW8 1/20 0.41
LMNA P02545 1/20 0.40
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39
TSHR P16473 1/20 0.39
KMT2A Q03164 1/20 0.39
HSD17B10 Q99714 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13634536 0.85 RAB9A (0.60) RAB9ASMN1; SMN2CHEK1KDM4EHDAC3
SCHEMBL13638811 0.81 RAB9A (0.63) RAB9ASMN1; SMN2CHEK1KDM4EHDAC3
SCHEMBL2771222 0.77 RAB9A (0.60) RAB9ASMN1; SMN2CHEK1KDM4EHDAC3
SCHEMBL14207028 0.74 CHEK1 (0.59) RAB9ASMN1; SMN2CHEK1KDM4EHDAC3
SCHEMBL14328610 0.74 RAB9A (0.54) RAB9ASMN1; SMN2CHEK1KDM4EHDAC3
SCHEMBL14207144 0.73 CHEK1 (0.83) RAB9ASMN1; SMN2CHEK1LMNAMAPT
SCHEMBL14207146 0.72 CHEK1 (0.81) RAB9ASMN1; SMN2CHEK1LMNAMAPT
SCHEMBL14207142 0.72 CHEK1 (0.81) RAB9ASMN1; SMN2CHEK1LMNAMAPT
SCHEMBL14328572 0.72 CHEK1 (0.64) RAB9ASMN1; SMN2CHEK1KDM4EIRAK4
SCHEMBL14207147 0.72 CHEK1 (0.64) RAB9ASMN1; SMN2CHEK1KDM4EHDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2078003-B1 ANILINOPIPERAZINE DERIVATIVES AND METHODS OF USE THEREOF MERCK SHARP & DOHME (US) 2017-03-08 EP disclosed