SCHEMBL186027

SCHEMBL186027

COc1cccc2[nH]nc(NS(=O)(=O)c3cccs3)c12

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.55
TP53 P04637 1/20 0.49
KDM4E B2RXH2 5/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
POLB P06746 1/20 0.48
KMT2A Q03164 4/20 0.47
MAPT P10636 3/20 0.47
MEN1 O00255 3/20 0.47
HTT P42858 2/20 0.47
TNF P01375 1/20 0.47
LMNA P02545 1/20 0.47
NOD2 Q9HC29 1/20 0.47
NOD1 Q9Y239 1/20 0.47
CCR4 P51679 1/20 0.47
LRRK2 Q5S007 1/20 0.45
GLA P06280 1/20 0.43
HPGD P15428 1/20 0.43
HSD17B10 Q99714 1/20 0.43
TTK P33981 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL250545 0.82 CCR4 (0.56) SMN1; SMN2KMT2AMEN1CCR4
SCHEMBL4740564 0.76 SMN1; SMN2 (0.56) ALDH1A1TP53KDM4ESMN1; SMN2POLB
SCHEMBL7571186 0.72 ALDH1A1 (1.00) ALDH1A1TP53KDM4ESMN1; SMN2POLB
SCHEMBL186310 0.70 CCR4 (0.73) ALDH1A1CCR4
SCHEMBL6180658 0.70 CCR4 (0.69) ALDH1A1TP53KDM4ESMN1; SMN2POLB
SCHEMBL186060 0.69 CCR4 (0.75) CCR4
SCHEMBL6180252 0.68 CCR4 (0.66) ALDH1A1TP53KDM4ESMN1; SMN2POLB
SCHEMBL15009538 0.68 ALDH1A1 (0.63) ALDH1A1TP53KDM4ESMN1; SMN2POLB
SCHEMBL4682088 0.67 KDM4E (0.67) ALDH1A1TP53KDM4ESMN1; SMN2POLB
SCHEMBL186026 0.66 TTK (0.60) ALDH1A1KDM4EPOLBKMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401270-A1 PYRAZOLE DERIVATIVES USED AS CCR4 RECEPTOR ANTAGONISTS Glaxo Group Limited (GB) 2012-01-04 EP disclosed