SCHEMBL18606705

SCHEMBL18606705

NS(=O)(=O)c1ccc(NC(=S)NC(=O)c2ccccc2[N+](=O)[O-])cc1

nearest known ligand 0.72

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA1 P00915 5/20 0.69
CA2 P00918 5/20 0.69
CA9 Q16790 5/20 0.69
ALDH1A1 P00352 7/20 0.66
KMT2A Q03164 6/20 0.66
MEN1 O00255 5/20 0.66
LMNA P02545 1/20 0.65
TDP1 Q9NUW8 2/20 0.64
MAPT P10636 2/20 0.64
PLK1 P53350 1/20 0.64
GAA P10253 2/20 0.60
ALPL P05186 2/20 0.60
HPGD P15428 1/20 0.60
L3MBTL1 Q9Y468 2/20 0.59
THRB P10828 1/20 0.59
KDM4E B2RXH2 1/20 0.57
ALPI P09923 1/20 0.57
ALPG P10696 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13454591 0.85 ALDH1A1 (0.65) ALDH1A1KMT2AMEN1LMNATDP1
SCHEMBL18606688 0.84 CA1 (0.74) CA1CA2CA9ALDH1A1LMNA
SCHEMBL13454491 0.82 LMNA (0.60) ALDH1A1KMT2AMEN1LMNATDP1
SCHEMBL12904257 0.82 ALDH1A1 (0.74) ALDH1A1KMT2AMEN1LMNATDP1
SCHEMBL18606689 0.81 CA1 (0.73) CA1CA2CA9ALDH1A1KMT2A
SCHEMBL13454744 0.81 LMNA (0.62) ALDH1A1KMT2AMEN1LMNATDP1
SCHEMBL13454617 0.80 POLB (0.59) ALDH1A1KMT2AMEN1LMNATDP1
SCHEMBL13454742 0.80 MAPT (0.61) CA1CA2CA9ALDH1A1KMT2A
SCHEMBL13453704 0.79 POLB (0.81) ALDH1A1KMT2AMEN1LMNAGAA
SCHEMBL13454664 0.79 ALDH1A1 (0.65) ALDH1A1KMT2AMEN1LMNATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170073306-A1 POTENT INHIBITORS OF HUMAN CARBONIC ANHYDRASE II AND BOVINE CARBONIC ANHYDRASE II AND THEIR MECHANISM OF ACTION CHOUDHARY MUHAMMAD IQBAL (PK) 2017-03-16 US claimed
US-20170073306-A1 POTENT INHIBITORS OF HUMAN CARBONIC ANHYDRASE II AND BOVINE CARBONIC ANHYDRASE II AND THEIR MECHANISM OF ACTION CHOUDHARY MUHAMMAD IQBAL (PK) 2017-03-16 US disclosed