SCHEMBL18616978

SCHEMBL18616978

O=C(NC1CCC1)c1cc(-c2ccc(F)c(F)c2)on1

nearest known ligand 0.73

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 12/20 0.73
RAB9A P51151 11/20 0.73
TDP1 Q9NUW8 1/20 0.73
MLLT1 Q03111 5/20 0.67
KMT2A Q03164 3/20 0.67
MEN1 O00255 2/20 0.67
TRPV1 Q8NER1 1/20 0.65
S1PR1 P21453 2/20 0.65
MLLT3 P42568 2/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17661429 0.85 NPC1 (1.00) NPC1RAB9ATDP1MLLT1KMT2A
SCHEMBL18618367 0.83 MLLT1 (0.95) NPC1RAB9ATDP1MLLT1KMT2A
SCHEMBL11931680 0.82 NPC1 (1.00) NPC1RAB9ATDP1MLLT1KMT2A
SCHEMBL17933816 0.82 NPC1 (0.95) NPC1RAB9ATDP1MLLT1KMT2A
SCHEMBL18617086 0.80 ACKR3 (0.74) NPC1RAB9ATDP1MLLT1KMT2A
SCHEMBL11931686 0.80 NPC1 (1.00) NPC1RAB9ATDP1MLLT1KMT2A
SCHEMBL11937745 0.79 TRPV1 (1.00) NPC1RAB9ATDP1MLLT1KMT2A
SCHEMBL17117167 0.79 NPC1 (1.00) NPC1RAB9ATDP1MLLT1KMT2A
SCHEMBL19245571 0.79 ROCK2 (0.57) NPC1RAB9ATDP1KMT2AMEN1
SCHEMBL13902147 0.78 S1PR1 (1.00) NPC1RAB9ATDP1MLLT1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017040606-A1 ISOXAZOLE DERIVATIVES FOR USE IN THE TREATMENT OF PULMONARY DISEASES AND DISORDERS PROTEOSTASIS THERAPEUTICS, INC. (US) 2017-03-09 WO disclosed