SCHEMBL18618367

SCHEMBL18618367

O=C(NC1CCC1)c1cc(-c2ccc(O)cc2)on1

nearest known ligand 0.95

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MLLT1 Q03111 5/20 0.95
NPC1 O15118 11/20 0.92
RAB9A P51151 10/20 0.92
KMT2A Q03164 4/20 0.92
TDP1 Q9NUW8 1/20 0.74
MEN1 O00255 3/20 0.73
S1PR1 P21453 2/20 0.73
MLLT3 P42568 2/20 0.71
TRPV1 Q8NER1 1/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17933816 0.88 NPC1 (0.95) MLLT1NPC1RAB9AKMT2ATDP1
SCHEMBL17661429 0.85 NPC1 (1.00) MLLT1NPC1RAB9AKMT2ATDP1
SCHEMBL11931680 0.85 NPC1 (1.00) MLLT1NPC1RAB9AKMT2ATDP1
SCHEMBL11931686 0.85 NPC1 (1.00) MLLT1NPC1RAB9AKMT2ATDP1
SCHEMBL13902147 0.84 S1PR1 (1.00) MLLT1NPC1RAB9AKMT2ATDP1
SCHEMBL18616978 0.83 NPC1 (0.73) MLLT1NPC1RAB9AKMT2ATDP1
SCHEMBL15099490 0.82 NPC1 (0.90) MLLT1NPC1RAB9AKMT2ATDP1
SCHEMBL11937745 0.82 TRPV1 (1.00) MLLT1NPC1RAB9AKMT2ATDP1
SCHEMBL14160551 0.79 TRPV1 (0.70) MLLT1NPC1RAB9AKMT2ATDP1
SCHEMBL16373728 0.77 NPC1 (0.81) MLLT1NPC1RAB9AKMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017040606-A1 ISOXAZOLE DERIVATIVES FOR USE IN THE TREATMENT OF PULMONARY DISEASES AND DISORDERS PROTEOSTASIS THERAPEUTICS, INC. (US) 2017-03-09 WO disclosed