SCHEMBL18636734

SCHEMBL18636734

CC(C)(C)OC(=O)NC1CN(c2cc(Cl)nc(N)n2)C1

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.53
AURKA O14965 6/20 0.52
PDPK1 O15530 6/20 0.52
AURKB Q96GD4 6/20 0.52
BTK Q06187 2/20 0.46
JAK3 P52333 1/20 0.46
MAP4K4 O95819 2/20 0.46
PDE10A Q9Y233 1/20 0.45
HSP90AA1 P07900 1/20 0.42
HSP90AB1 P08238 1/20 0.42
HRH3 Q9Y5N1 1/20 0.42
HRH4 Q9H3N8 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
MAPT P10636 1/20 0.42
SUV39H2 Q9H5I1 2/20 0.42
EIF2AK4 Q9P2K8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12119818 0.91 AURKA (0.63) LMNAAURKAPDPK1AURKBBTK
SCHEMBL31741685 0.91 LMNA (0.57) LMNAAURKAPDPK1AURKBBTK
SCHEMBL16977369 0.89 AURKA (0.63) LMNAAURKAPDPK1AURKBBTK
SCHEMBL12118769 0.89 AURKA (0.63) LMNAAURKAPDPK1AURKBBTK
SCHEMBL27717380 0.88 LMNA (0.60) LMNAAURKAPDPK1AURKBHRH3
SCHEMBL27738450 0.83 LMNA (0.53) LMNAPDE10AHRH3HRH4CYP1A2
SCHEMBL18636729 0.83 HRH4 (0.55) AURKAPDPK1AURKBBTKJAK3
SCHEMBL12119179 0.82 AURKA (0.63) LMNAAURKAPDPK1AURKBBTK
SCHEMBL12119518 0.82 AURKA (0.63) LMNAAURKAPDPK1AURKBBTK
SCHEMBL3196818 0.82 LMNA (0.56) LMNAHRH3HRH4CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1966162-B1 PYRIMIDINE DERIVATIVES ZIARCO PHARMA LTD (GB) 2017-03-15 EP disclosed