SCHEMBL18638342

SCHEMBL18638342

CC(C)(O)CN1CNc2cc(-c3ccc(C(F)(F)F)cc3)ccc21

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 7/20 0.36
MCHR1 Q99705 1/20 0.35
CYP3A4 P08684 1/20 0.34
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33
MARS1 P56192 1/20 0.33
APP P05067 1/20 0.33
TDP2 O95551 1/20 0.33
BRD4 O60885 1/20 0.32
BRD2 P25440 1/20 0.32
BRD3 Q15059 1/20 0.32
SIGMAR1 Q99720 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32
CHKA P35790 1/20 0.32
AGXT P21549 1/20 0.32
NISCH Q9Y2I1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18638540 0.90 KIF11 (0.39) KIF11MCHR1CYP3A4MEN1GAA
SCHEMBL18638653 0.89 PARP10 (0.38) KIF11MAPTHRH3
SCHEMBL18638664 0.87 APP (0.42) APP
SCHEMBL18638652 0.85 GRM2 (0.36) KDM4EMEN1GAAMAPTKMT2A
SCHEMBL18638669 0.84 ABL1 (0.40) MCHR1HRH3NISCH
SCHEMBL20393281 0.80 PARP10 (0.38) KIF11MAPTHRH3
SCHEMBL18638666 0.79
SCHEMBL18638655 0.79 PGR (0.41)
SCHEMBL20393147 0.78 APP (0.42) APP
SCHEMBL18638339 0.76 FASN (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017043636-A1 NOVEL BENZIMIDAZOLE COMPOUND AND PHARMACEUTICAL USE OF SAME 大日本住友製薬株式会社 2017-03-16 WO disclosed