SCHEMBL18640100

SCHEMBL18640100

Nc1n[nH]c2cc(OCc3ccc(C(F)(F)F)cc3)ccc12

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MAOB P27338 13/20 0.56
MAOA P21397 5/20 0.49
AR P10275 1/20 0.48
PPARD Q03181 2/20 0.44
PPARA Q07869 2/20 0.44
PPARG P37231 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13736416 0.89 KIT (0.54) MAOB
SCHEMBL18639944 0.83 MAOB (0.47) MAOBMAOAAR
SCHEMBL18639883 0.83 MAOB (0.49) MAOBMAOAAR
SCHEMBL18640073 0.83 IKBKE (0.43) MAOA
SCHEMBL216014 0.83 CNR2 (0.54) MAOB
SCHEMBL11963403 0.82 IKBKE (0.54) MAOBMAOA
SCHEMBL18639882 0.80 MAOA (0.50) MAOBMAOAAR
SCHEMBL18640122 0.78 CYP2D6 (0.51) MAOBMAOA
SCHEMBL18639861 0.78 MAPK1 (0.50) MAOBMAOA
SCHEMBL13736786 0.77 KIT (0.55) MAOBMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017045751-A1 COMPOUNDS AS ASIC INHIBITORS AND USES THEREOF MERCK PATENT GMBH (DE) 2017-03-23 WO disclosed
WO-2017045751-A1 COMPOUNDS AS ASIC INHIBITORS AND USES THEREOF MERCK PATENT GMBH (DE) 2017-03-23 WO disclosed