SCHEMBL186441

SCHEMBL186441

COc1ccc(Nc2ccc(N)cc2C)c(C)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.60
ADRA2A P08913 1/20 0.53
ADRA2C P18825 1/20 0.53
ADRA1D P25100 1/20 0.53
ADRA1A P35348 1/20 0.53
ADRA1B P35368 1/20 0.53
NR4A1 P22736 1/20 0.47
TDP1 Q9NUW8 2/20 0.47
MAPK1 P28482 1/20 0.47
ALDH1A1 P00352 3/20 0.46
CYP3A4 P08684 2/20 0.46
FLT3 P36888 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.43
RAB9A P51151 1/20 0.42
OPRM1 P35372 1/20 0.42
CA12 O43570 2/20 0.42
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
CA9 Q16790 2/20 0.42
SIGMAR1 Q99720 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL186343 0.86 NR4A1 (0.62) GAANR4A1TDP1MAPK1ALDH1A1
SCHEMBL4230288 0.81 GAA (0.64) GAAADRA2AADRA2CADRA1DADRA1A
SCHEMBL11219654 0.81 GAA (0.64) GAAADRA2AADRA2CADRA1DADRA1A
SCHEMBL6439831 0.81 GAA (0.64) GAAADRA2AADRA2CADRA1DADRA1A
Hydrochloric Acid SCHEMBL6438214 0.80 MAPT (0.62) GAAADRA2AADRA2CADRA1DADRA1A
SCHEMBL10639862 0.80 GAA (0.72) GAAADRA2AADRA2CADRA1DADRA1A
SCHEMBL25634740 0.78 GAA (0.80) GAAADRA2AADRA2CADRA1DADRA1A
SCHEMBL10640322 0.77 GAA (0.58) GAAADRA2AADRA2CADRA1DADRA1A
SCHEMBL4791618 0.77 GAA (0.58) GAAADRA2AADRA2CADRA1DADRA1A
SCHEMBL15698752 0.77 ADRA2A (0.51) GAAADRA2AADRA2CADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401256-A1 COMPOUNDS AS BRADYKININ B1 ANTAGONISTS Boehringer Ingelheim International GmbH (DE) 2012-01-04 EP disclosed
WO-2010097372-A1 COMPOUNDS AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed