SCHEMBL186343

SCHEMBL186343

COc1ccc(Nc2ccc(N)cc2C)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A1 P22736 1/20 0.62
GAA P10253 4/20 0.61
ALDH1A1 P00352 6/20 0.53
TDP1 Q9NUW8 5/20 0.53
MAPT P10636 5/20 0.53
RAB9A P51151 4/20 0.53
KDM4E B2RXH2 3/20 0.53
THRB P10828 2/20 0.53
RECQL P46063 2/20 0.53
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
HTT P42858 1/20 0.53
MMP14 P50281 1/20 0.53
MAPK1 P28482 5/20 0.52
L3MBTL1 Q9Y468 3/20 0.52
NPC1 O15118 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
CYP3A4 P08684 1/20 0.47
LMNA P02545 2/20 0.46
POLB P06746 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL186441 0.86 GAA (0.60) NR4A1GAAALDH1A1TDP1MAPT
SCHEMBL25634740 0.86 GAA (0.80) NR4A1GAAALDH1A1TDP1MAPT
SCHEMBL9629642 0.83 GAA (0.65) GAAALDH1A1TDP1MAPTRAB9A
SCHEMBL21131527 0.80 GAA (0.61) NR4A1GAAALDH1A1TDP1MAPT
SCHEMBL11555581 0.80 GAA (0.61) GAAALDH1A1TDP1MAPTRAB9A
SCHEMBL29764005 0.80 ALDH1A1 (0.50) GAAALDH1A1TDP1MAPTKDM4E
SCHEMBL29595 0.80 ALDH1A1 (0.50) GAAALDH1A1TDP1MAPTKDM4E
SCHEMBL2952972 0.79 GAA (0.75) GAAALDH1A1TDP1MAPTRAB9A
SCHEMBL6999192 0.79 GAA (0.75) GAAALDH1A1TDP1MAPTRAB9A
SCHEMBL11206431 0.79 GAA (0.65) GAAALDH1A1TDP1MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401256-A1 COMPOUNDS AS BRADYKININ B1 ANTAGONISTS Boehringer Ingelheim International GmbH (DE) 2012-01-04 EP disclosed
WO-2010097372-A1 COMPOUNDS AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed