SCHEMBL1864563

SCHEMBL1864563

CC(C)(C)N(C(=O)O)C1CCN(C2CCC(Cl)(Cl)CC2)CC1

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.33
TACR1 P25103 4/20 0.32
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
KMT2A Q03164 1/20 0.31
KCNH2 Q12809 2/20 0.31
CCR5 P51681 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1306189 0.86 ALDH1A1 (0.35) MEN1ALDH1A1KMT2AKCNH2CCR5
SCHEMBL988772 0.83 ALDH1A1 (0.39) MEN1ALDH1A1KMT2AKCNH2CCR5
SCHEMBL1306995 0.83 ALDH1A1 (0.42) MEN1ALDH1A1KMT2AKCNH2
SCHEMBL4939731 0.79 HRH3 (0.37) ALDH1A1
SCHEMBL16633564 0.78 CCR5 (0.32) MEN1ALDH1A1KMT2ACCR5
SCHEMBL28851402 0.78 HTR2A (0.31) MEN1ALDH1A1KMT2A
SCHEMBL1307534 0.77 CCR5 (0.35) MEN1ALDH1A1KMT2AKCNH2CCR5
SCHEMBL16372187 0.77 OPRL1 (0.34)
SCHEMBL600511 0.77 ACACB (0.32) MEN1ALDH1A1KMT2ACCR5
SCHEMBL2694217 0.76 MEN1 (0.38) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011006794-A9 3-OXO-2, 3-DIHYDRO-1H-ISOINDOLE-4-CARBOXAMIDES AS PARP INHIBITORS NERVIANO MEDICAL SCIENCES S.R.L. (IT) 2011-05-05 WO disclosed