SCHEMBL18652292

SCHEMBL18652292

Cn1ncc2cc(-c3cccc(N)c3)ccc21

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 5/20 0.51
TRPA1 O75762 1/20 0.51
MAP4K4 O95819 2/20 0.46
FAAH O00519 1/20 0.45
SRC P12931 2/20 0.44
USP7 Q93009 1/20 0.44
AR P10275 3/20 0.44
APP P05067 1/20 0.44
MEN1 O00255 1/20 0.44
PSIP1 O75475 1/20 0.44
AXL P30530 1/20 0.44
MKNK1 Q9BUB5 1/20 0.44
MKNK2 Q9HBH9 1/20 0.44
NR3C1 P04150 1/20 0.43
MAOA P21397 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23638931 0.83 TRPA1 (0.60) TRPA1FAAHSRCUSP7AR
SCHEMBL13680579 0.83 NR3C1 (0.60) TRPA1FAAHARAPPNR3C1
SCHEMBL378619 0.81 CHEK1 (0.57) TRPA1SRCUSP7ARAPP
SCHEMBL30006507 0.81 CHEK1 (0.57) TRPA1SRCUSP7ARAPP
SCHEMBL20004068 0.81 TRPA1 (0.55) TRPA1FAAHARAPPNR3C1
SCHEMBL5343977 0.80 CHEK1 (0.56) TRPA1SRCUSP7ARAPP
SCHEMBL17547028 0.79 TRPA1 (0.49) TRPA1FAAHUSP7ARAPP
SCHEMBL15340863 0.79 TRPA1 (0.49) IRAK4TRPA1FAAHARAPP
SCHEMBL21464284 0.78 TRPA1 (0.58) TRPA1FAAHSRCUSP7AR
SCHEMBL31729795 0.77 TRPA1 (0.54) TRPA1FAAHSRCUSP7AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3144311-A1 TRICYCLIC HETEROCYCLIC DERIVATIVE HAVING HIV REPLICATION-INHIBITING EFFECT Shionogi & Co., Ltd. (JP) 2017-03-22 EP disclosed