SCHEMBL1866587

SCHEMBL1866587

O=C(O)N1CCC(=Cc2cccc(F)c2[N+](=O)[O-])CC1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 6/20 0.40
LMNA P02545 4/20 0.38
POLB P06746 3/20 0.35
ALDH1A1 P00352 4/20 0.34
MAPT P10636 2/20 0.34
NTSR1 P30989 1/20 0.34
GAA P10253 2/20 0.34
CASP3 P42574 1/20 0.33
USP14 P54578 1/20 0.33
UCHL5 Q9Y5K5 1/20 0.33
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
CES2 O00748 1/20 0.33
CES1 P23141 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.32
MAPK1 P28482 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22556714 0.79 TSHR (0.47) LMNAPOLBALDH1A1MAPTKMT2A
SCHEMBL1865742 0.77 SRD5A2 (0.41) SRD5A2LMNAALDH1A1MAPTGAA
SCHEMBL22556898 0.75 MAPT (0.39) SRD5A2LMNAALDH1A1MAPTGAA
SCHEMBL1872138 0.74 CASP3 (0.39) SRD5A2LMNAALDH1A1MAPTGAA
SCHEMBL1863164 0.72 CASP3 (0.47) SRD5A2LMNAPOLBALDH1A1MAPT
SCHEMBL1862784 0.72 ACHE (0.51) LMNAALDH1A1MAPTKMT2AMEN1
SCHEMBL15537076 0.71 SRD5A2 (0.51) SRD5A2ALDH1A1MAPTKMT2A
SCHEMBL1870246 0.70 CASP3 (0.47) SRD5A2LMNAALDH1A1MAPTGAA
SCHEMBL16950618 0.70 MEN1 (0.45) LMNAPOLBALDH1A1MAPTNTSR1
SCHEMBL27140785 0.70 MAPT (0.58) LMNAPOLBALDH1A1MAPTNTSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2493855-A1 (1,1, 1,3, 3, 3-HEXAFLUORO-2-HYDROXYPROPAN-2-YL) PHENYL DERIVATIVES, PHARMACEUTICAL COMPOSITIONS THEREOF AND THEIR USE FOR THE TREATMENT OF ATHEROSCLEROSIS MSD Oss B.V. (NL) 2012-09-05 EP disclosed
WO-2011051282-A1 (1,1, 1,3, 3, 3-HEXAFLUORO-2-HYDROXYPROPAN-2-YL) PHENYL DERIVATIVES, PHARMACEUTICAL COMPOSITIONS THEREOF AND THEIR USE FOR THE TREATMENT OF ATHEROSCLEROSIS N.V. ORGANON (NL) 2011-05-05 WO disclosed