SCHEMBL1866735

SCHEMBL1866735

NC1CN(c2ccc(-c3cccnc3)cc2)C1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 3/20 0.48
ALDH1A1 P00352 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
APP P05067 1/20 0.46
MKNK1 Q9BUB5 3/20 0.45
MKNK2 Q9HBH9 3/20 0.45
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA9 Q16790 1/20 0.45
KDM1A O60341 1/20 0.45
MAOA P21397 1/20 0.45
MAOB P27338 1/20 0.45
KIF11 P52732 1/20 0.44
CYP11B2 P19099 1/20 0.44
CHRNB2 P17787 2/20 0.43
CHRNA4 P43681 2/20 0.43
NAAA Q02083 1/20 0.42
CHRNA7 P36544 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30608959 0.81 CHRNB2 (0.62) CHRNB2CHRNA4CHRNA7
SCHEMBL16515661 0.81 CHRNB2 (0.62) CHRNB2CHRNA4CHRNA7
SCHEMBL928568 0.80 CHRNB2 (0.55) CYP2A6ALDH1A1CYP1A2CYP3A4APP
SCHEMBL930530 0.80 CHRNB2 (0.68) CHRNB2CHRNA4CHRNA7
SCHEMBL1865509 0.78 CYP2A6 (0.54) CYP2A6ALDH1A1CYP1A2CYP3A4APP
SCHEMBL928620 0.77 HRH3 (0.58) APPKIF11CHRNB2CHRNA4CHRNA7
SCHEMBL1791787 0.77 CHRNB2 (0.72) CHRNB2CHRNA4CHRNA7
SCHEMBL1794946 0.77 HRH3 (0.58) APPKIF11CHRNB2CHRNA4CHRNA7
SCHEMBL930536 0.77 CHRNB2 (0.72) CHRNB2CHRNA4CHRNA7
SCHEMBL1863933 0.77 ALDH1A1 (0.52) CYP2A6ALDH1A1CYP1A2CYP3A4APP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011053705-A1 PYRIMIDINE COMPOUNDS AS DELTA OPIOID RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2011-05-05 WO disclosed