SCHEMBL18667635

SCHEMBL18667635

CN(C)CCCOc1ccc(-c2ncc(CNC(=O)c3ccc4c(c3Cl)NC(=O)c3ccccc3S4)s2)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 2/20 0.35
ROCK1 Q13464 2/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
TP53 P04637 5/20 0.34
MAPT P10636 4/20 0.34
LMNA P02545 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
CHEK1 O14757 1/20 0.33
NAMPT P43490 1/20 0.33
POLB P06746 2/20 0.33
LSS P48449 1/20 0.33
USP7 Q93009 1/20 0.33
USP47 Q96K76 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
CXCR1 P25024 2/20 0.33
PARP1 P09874 1/20 0.32
MAOB P27338 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18667107 0.92 ROCK2 (0.36) ROCK2ROCK1CYP3A4CYP2D6CYP2C9
SCHEMBL18667628 0.87 ROCK2 (0.34) ROCK2ROCK1CYP3A4CYP2D6CYP2C9
SCHEMBL21250468 0.86 ROCK2 (0.34) ROCK2ROCK1CYP3A4CYP2D6CYP2C9
SCHEMBL19984576 0.84 ROCK2 (0.38) ROCK2ROCK1CYP3A4CYP2D6CYP2C9
SCHEMBL18667626 0.81 HDAC1 (0.37) ROCK2ROCK1CYP3A4CYP2D6CYP2C9
SCHEMBL21250432 0.81 RXFP1 (0.45) ROCK2ROCK1TP53MAPTMEN1
SCHEMBL18667142 0.81 ROCK2 (0.35) ROCK2ROCK1CYP3A4CYP2D6CYP2C9
SCHEMBL21250368 0.80 ROCK2 (0.34) ROCK2ROCK1CYP3A4CYP2D6CYP2C9
SCHEMBL18667750 0.79 NAMPT (0.36) TP53MAPTNAMPTPOLBRXFP1
SCHEMBL23018413 0.78 KMT2A (0.45) TP53MAPTMEN1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017048950-A1 HEPATITIS B CORE PROTEIN MODULATORS ASSEMBLY BIOSCIENCES, INC. (US) 2017-03-23 WO disclosed