SCHEMBL19984576

SCHEMBL19984576

Cc1c(C(=O)NCc2cnc(-c3ccc(OCCCN(C)C)cc3)s2)ccc2c1NC(=O)c1ccncc1S2

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
ROCK1 Q13464 1/20 0.38
HRH3 Q9Y5N1 1/20 0.33
CHEK1 O14757 1/20 0.33
EED O75530 1/20 0.33
SUZ12 Q15022 1/20 0.33
EZH2 Q15910 1/20 0.33
PARP1 P09874 1/20 0.32
LMNA P02545 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
LTA4H P09960 1/20 0.32
NAMPT P43490 1/20 0.31
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18667107 0.91 ROCK2 (0.36) ROCK2CYP3A4CYP2D6CYP2C9ROCK1
SCHEMBL24221908 0.89 ROCK2 (0.37) ROCK2CYP3A4CYP2D6CYP2C9ROCK1
SCHEMBL21291434 0.86 ROCK2 (0.36) ROCK2CYP3A4CYP2D6CYP2C9ROCK1
SCHEMBL18667635 0.84 ROCK2 (0.35) ROCK2CYP3A4CYP2D6CYP2C9ROCK1
SCHEMBL18667626 0.82 HDAC1 (0.37) ROCK2CYP3A4CYP2D6CYP2C9ROCK1
SCHEMBL18667142 0.82 ROCK2 (0.35) ROCK2CYP3A4CYP2D6CYP2C9ROCK1
SCHEMBL21250368 0.81 ROCK2 (0.34) ROCK2CYP3A4CYP2D6CYP2C9ROCK1
SCHEMBL18667750 0.78 NAMPT (0.36) SMN1; SMN2NAMPT
SCHEMBL19984640 0.78 SLC22A12 (0.35) ROCK2
SCHEMBL18667628 0.76 ROCK2 (0.34) ROCK2CYP3A4CYP2D6CYP2C9ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018053157-A1 HEPATITIS B CORE PROTEIN MODULATORS ASSEMBLY BIOSCIENCES, INC. (US) 2018-03-22 WO disclosed