SCHEMBL18668657

SCHEMBL18668657

O=C(O)NCc1ccc(C(=O)Nc2cccc3cccnc23)cc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 4/20 0.70
HDAC6 Q9UBN7 4/20 0.67
L3MBTL1 Q9Y468 2/20 0.65
TDP1 Q9NUW8 1/20 0.65
GAA P10253 1/20 0.65
HDAC3 O15379 3/20 0.65
HDAC1 Q13547 3/20 0.65
HDAC2 Q92769 3/20 0.65
HDAC4 P56524 1/20 0.63
HDAC7 Q8WUI4 1/20 0.63
HDAC10 Q969S8 1/20 0.63
HDAC11 Q96DB2 1/20 0.63
HDAC8 Q9BY41 1/20 0.63
HDAC9 Q9UKV0 1/20 0.63
HDAC5 Q9UQL6 1/20 0.63
NCOR2 Q9Y618 1/20 0.63
KMT2A Q03164 2/20 0.62
POLB P06746 1/20 0.62
MAPT P10636 4/20 0.61
NPC1 O15118 2/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24522646 0.88 HDAC6 (0.74) KDRHDAC6L3MBTL1TDP1GAA
SCHEMBL18668729 0.87 HDAC6 (0.62) KDRHDAC6L3MBTL1TDP1GAA
SCHEMBL18668668 0.85 HDAC6 (0.73) KDRHDAC6L3MBTL1TDP1GAA
SCHEMBL16456367 0.84 POLB (0.73) KDRHDAC6L3MBTL1TDP1GAA
SCHEMBL18688205 0.83 NAMPT (0.61) KDRHDAC6L3MBTL1TDP1GAA
SCHEMBL6260903 0.83 KDR (1.00) KDRHDAC6L3MBTL1TDP1GAA
SCHEMBL29434873 0.83 KDR (1.00) KDRHDAC6L3MBTL1TDP1GAA
SCHEMBL15441206 0.82 KDR (0.77) KDRHDAC6L3MBTL1TDP1GAA
SCHEMBL15093487 0.82 HDAC6 (0.77) KDRHDAC6L3MBTL1TDP1GAA
SCHEMBL16456332 0.82 HDAC6 (0.77) KDRHDAC6L3MBTL1TDP1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017053360-A1 BICYCLIC AND TRICYCLIC CAP BEARING MERCAPTOACETAMIDE DERIVATIVES AS HISTONE DEACETYLASE INHIBITORS THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2017-03-30 WO disclosed