SCHEMBL18669448

SCHEMBL18669448

COc1nc(OC2CCC(F)CC2)c(F)cc1C#N

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.36
ACACB O00763 7/20 0.36
NSD2 O96028 1/20 0.35
GPR6 P46095 2/20 0.34
KDM4E B2RXH2 4/20 0.33
MEN1 O00255 2/20 0.33
ALDH1A1 P00352 2/20 0.33
KMT2A Q03164 2/20 0.33
DCK P27707 1/20 0.33
POLB P06746 2/20 0.32
HPGD P15428 1/20 0.32
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32
PIK3CA P42336 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18669574 0.91 GAA (0.37) GAAACACBNSD2GPR6KDM4E
SCHEMBL18669555 0.85 GAA (0.35) GAAACACBNSD2GPR6KDM4E
SCHEMBL18669614 0.77 KHK (0.47) GAAACACBNSD2KDM4EALDH1A1
SCHEMBL18669540 0.76 ACACB (0.36) ACACBNSD2GPR6
SCHEMBL20510904 0.76 AR (0.40) GPR6KDM4EALDH1A1
SCHEMBL18669671 0.69 TBK1 (0.34) ACACB
SCHEMBL6186446 0.69 KHK (0.57) GAAKDM4EMEN1ALDH1A1KMT2A
SCHEMBL3622824 0.67 ROCK2 (0.46) GAANSD2KDM4EALDH1A1HPGD
SCHEMBL18669615 0.67 GRM1 (0.37) ACACBPIK3CA
SCHEMBL1937799 0.66 ROCK2 (0.63) GAANSD2KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3353155-A1 PYRIDYL OR PYRAZINYL COMPOUNDS CARRYING A METHYL-BOUND ALPHA-AMINO ACID AMIDE GROUP AbbVie Deutschland GmbH & Co. KG (DE) 2018-08-01 EP disclosed
WO-2017050807-A1 PYRIDYL OR PYRAZINYL COMPOUNDS CARRYING A METHYL-BOUND ALPHA-AMINO ACID AMIDE GROUP AbbVie Deutschland GmbH & Co. KG (DE) 2017-03-30 WO disclosed