SCHEMBL1867178

SCHEMBL1867178

CN(CC(NC(=O)OC(C)(C)C)C(Cc1ccccc1)C1CCCC1)C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KLK5 Q9Y337 3/20 0.49
ACE P12821 2/20 0.46
ATM Q13315 2/20 0.45
PSEN1 P49768 2/20 0.44
PSEN2 P49810 2/20 0.44
APH1B Q8WW43 2/20 0.44
NCSTN Q92542 2/20 0.44
APH1A Q96BI3 2/20 0.44
PSENEN Q9NZ42 2/20 0.44
CTSS P25774 2/20 0.43
CTSL P07711 1/20 0.43
CTSB P07858 1/20 0.43
CTSK P43235 1/20 0.43
KMT2A Q03164 2/20 0.43
REN P00797 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1859578 0.92 KLK5 (0.45) KLK5ACEATMPSEN1PSEN2
SCHEMBL1859576 0.92 KLK5 (0.45) KLK5ACEATMPSEN1PSEN2
SCHEMBL1861663 0.91 KLK5 (0.45) KLK5ACEATMPSEN1PSEN2
SCHEMBL1861665 0.91 KLK5 (0.45) KLK5ACEATMPSEN1PSEN2
SCHEMBL1861930 0.85 KLK5 (0.43) KLK5ACEATMPSEN1PSEN2
SCHEMBL7356966 0.79 KLK5 (0.59) KLK5ACEATMCTSSCTSL
SCHEMBL498943 0.76 HTR2C (0.38) KLK5ACEATMCTSLKMT2A
SCHEMBL1864930 0.76 ATM (0.46) KLK5ACEATMCTSSCTSL
SCHEMBL1861190 0.76 L3MBTL1 (0.46) KMT2AL3MBTL1
SCHEMBL5222884 0.75 KLK5 (0.59) KLK5ATMPSEN1PSEN2APH1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110105506-A1 Diaminoalkane aspartic protease inhibitors VITAE PHARMACEUTICALS, INC. 2011-05-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110105506-A1 Diaminoalkane aspartic protease inhibitors DNPEP, PEPD, ACE KLK5 256/4885ACE 3/4885ATM 2336/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.