SCHEMBL498943

SCHEMBL498943

CN(CC(NC(=O)O)[C@H](Cc1ccccc1)[C@H]1CCCOC1)C(=O)OC(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.38
SLC6A4 P31645 1/20 0.38
ACE P12821 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
KMT2A Q03164 1/20 0.36
KLK5 Q9Y337 1/20 0.35
MLNR O43193 1/20 0.35
ABCB11 O95342 1/20 0.35
LMNA P02545 1/20 0.35
CTSD P07339 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP3A5 P20815 1/20 0.35
CNR1 P21554 1/20 0.35
TBXAS1 P24557 1/20 0.35
ADRA1A P35348 1/20 0.35
CTSL P07711 1/20 0.35
CCR5 P51681 1/20 0.34
ATM Q13315 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL499419 0.79 SMN1; SMN2 (0.38) MLNRABCB11LMNACTSDCYP3A4
SCHEMBL499681 0.79 SMN1; SMN2 (0.38) MLNRABCB11LMNACTSDCYP3A4
SCHEMBL1867178 0.76 KLK5 (0.49) ACEL3MBTL1KMT2AKLK5CTSL
SCHEMBL1861665 0.72 KLK5 (0.45) ACEKMT2AKLK5CTSLATM
SCHEMBL1861663 0.72 KLK5 (0.45) ACEKMT2AKLK5CTSLATM
SCHEMBL8110118 0.72 SYK (0.46) KMT2AKLK5LMNACYP3A4CTSL
SCHEMBL1859576 0.71 KLK5 (0.45) ACEKMT2AKLK5CTSLATM
SCHEMBL1859578 0.71 KLK5 (0.45) ACEKMT2AKLK5CTSLATM
SCHEMBL3002580 0.71 CTSS (0.34) HTR2CSLC6A4KMT2A
SCHEMBL498942 0.71 HTR2C (0.38) HTR2CSLC6A4L3MBTL1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8106221-B2 Renin inhibitors VITAE PHARMACEUTICALS, INC. (US) 2012-01-31 US disclosed