SCHEMBL1867434

SCHEMBL1867434

COC(=O)C1CC2C=CC=CC2=C2CCCNC21

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.34
CYP2D6 P10635 3/20 0.34
CYP1A2 P05177 2/20 0.34
CYP2C19 P33261 1/20 0.34
TSHR P16473 2/20 0.33
CYP2C9 P11712 1/20 0.33
MAPK1 P28482 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12493061 0.65 CHRNB2 (0.31)
Hydrochloric Acid SCHEMBL10912090 0.63
SCHEMBL2723936 0.63 CHRNB2 (0.31)
SCHEMBL4874913 0.61
SCHEMBL24179852 0.59 CYP3A4 (0.39) CYP3A4CYP2D6CYP1A2CYP2C19TSHR
SCHEMBL7654723 0.58 SLC6A2 (0.50) CYP3A4CYP2D6CYP1A2CYP2C19TSHR
SCHEMBL9294530 0.58 SLC6A2 (0.50) CYP3A4CYP2D6CYP1A2CYP2C19TSHR
SCHEMBL27298881 0.58 SLC6A2 (0.50) CYP3A4CYP2D6CYP1A2CYP2C19TSHR
SCHEMBL8494369 0.56 CHRM2 (0.48) CYP3A4CYP2D6CYP1A2CYP2C19TSHR
SCHEMBL974399 0.56 CHRM2 (0.48) CYP3A4CYP2D6CYP1A2CYP2C19TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2496559-A1 ARYL- AND HETEROARYLCARBONYL DERIVATIVES OF HEXAHYDROINDENOPYRIDINE AND OCTAHYDROBENZOQUINOLINE Vitae Pharmaceuticals, Inc. (US) 2012-09-12 EP disclosed
WO-2011057054-A1 ARYL- AND HETEROARYLCARBONYL DERIVATIVES OF HEXAHYDROINDENOPYRIDINE AND OCTAHYDROBENZOQUINOLINE VITAE PHARMACEUTICALS, INC. (US) 2011-05-12 WO disclosed