SCHEMBL1868192

SCHEMBL1868192

CC(C)Cc1ccc2ncccc2c1.CCCCc1ccc2ccccc2n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 2/20 0.42
CYSLTR1 Q9Y271 7/20 0.41
CYSLTR2 Q9NS75 6/20 0.41
GPBAR1 Q8TDU6 5/20 0.41
ALOX5AP P20292 2/20 0.41
TLR8 Q9NR97 1/20 0.39
MAPK1 P28482 2/20 0.39
ALDH1A1 P00352 2/20 0.39
TP53 P04637 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
TSHR P16473 1/20 0.39
NFKB1 P19838 1/20 0.39
CYP2C19 P33261 1/20 0.39
HIF1A Q16665 1/20 0.39
ACACB O00763 1/20 0.39
MEN1 O00255 1/20 0.39
GMNN O75496 1/20 0.39
LMNA P02545 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Quinoline SCHEMBL28839000 0.84 ALDH1A1 (0.53) PDE10ACYSLTR1CYSLTR2GPBAR1TLR8
SCHEMBL19182788 0.80 CYP1A2 (0.47) PDE10ACYSLTR1CYSLTR2GPBAR1ALOX5AP
SCHEMBL29873370 0.80 ALDH1A1 (0.53) PDE10AALDH1A1TP53TSHRACACB
SCHEMBL113636 0.80 ALDH1A1 (0.53) PDE10AALDH1A1TP53TSHRACACB
Quinoline SCHEMBL28287745 0.79 KCNH2 (0.51) PDE10ACYSLTR1CYSLTR2GPBAR1TLR8
SCHEMBL6115157 0.76 ALDH1A1 (0.51) PDE10AALDH1A1TP53TSHRSMN1; SMN2
SCHEMBL29827516 0.76 ALDH1A1 (0.51) PDE10AALDH1A1TP53TSHRSMN1; SMN2
SCHEMBL538491 0.76 GPBAR1 (0.54) PDE10ACYSLTR1CYSLTR2GPBAR1TLR8
SCHEMBL13034790 0.75 ALDH1A1 (0.53) PDE10AMAPK1ALDH1A1TP53CYP1A2
Hydrochloric Acid SCHEMBL27600363 0.75 GPBAR1 (0.52) PDE10ACYSLTR1CYSLTR2GPBAR1TLR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2496682-A1 DELIVERY PARTICLE The Procter & Gamble Company (US) 2012-09-12 EP disclosed
WO-2011056935-A1 DELIVERY PARTICLE THE PROCTER & GAMBLE COMPANY (US) 2011-05-12 WO disclosed