SCHEMBL1869009

SCHEMBL1869009

CCCn1c(Oc2cccc(OC)c2)nc(=O)c2c1N=C(C1CC=CC1)[N]2

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 5/20 0.47
ADORA3 P0DMS8 1/20 0.47
DRD2 P14416 3/20 0.38
ADORA2B P29275 1/20 0.37
ALPL P05186 1/20 0.36
MEN1 O00255 2/20 0.34
ALDH1A1 P00352 2/20 0.34
KMT2A Q03164 2/20 0.34
TSHR P16473 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
HIF1A Q16665 1/20 0.33
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1875007 0.90 ADORA1 (0.55) ADORA1ADORA3DRD2ADORA2BALPL
SCHEMBL1871179 0.89 ADORA1 (0.46) ADORA1ADORA3DRD2ADORA2BMEN1
SCHEMBL1871234 0.81 ADORA1 (0.47) ADORA1ADORA3DRD2ADORA2B
SCHEMBL1870359 0.79 ADORA1 (0.44) ADORA1ADORA3ADORA2BALPL
SCHEMBL1870513 0.79 ADORA1 (0.58) ADORA1ADORA3DRD2ADORA2B
SCHEMBL1866939 0.78 ADORA1 (0.44) ADORA1ADORA3ADORA2BALPL
SCHEMBL1864689 0.77 ADORA1 (0.44) ADORA1ADORA3ADORA2BSMN1; SMN2
SCHEMBL1870705 0.76 ADORA1 (0.42) ADORA1ADORA3ADORA2B
SCHEMBL1871420 0.75 ADORA1 (0.41) ADORA1ADORA3ADORA2BMEN1KMT2A
SCHEMBL1869240 0.74 ADORA1 (0.38) ADORA1ADORA3ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2499142-A1 SUBSTITUTED FUSED PYRIMIDINE COMPOUNDS, ITS PREPARATION AND USES THEREOF Advinus Therapeutics Limited (IN) 2012-09-19 EP disclosed
WO-2011055391-A1 SUBSTITUTED FUSED PYRIMIDINE COMPOUNDS, ITS PREPARATION AND USES THEREOF ADVINUS THERAPEUTICS PRIVATE LIMITED (IN) 2011-05-12 WO disclosed