SCHEMBL1870513

SCHEMBL1870513

CCCn1c(Oc2cccc(C(F)(F)F)c2)nc(=O)c2c1N=C(C1CCCCC1)[N]2

nearest known ligand 0.58

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 9/20 0.58
ADORA3 P0DMS8 1/20 0.44
DRD2 P14416 1/20 0.38
ADORA2B P29275 1/20 0.36
CTSK P43235 1/20 0.35
UBE2M P61081 1/20 0.34
DCUN1D1 Q96GG9 1/20 0.34
FFAR4 Q5NUL3 1/20 0.34
LTA4H P09960 1/20 0.34
MAPT P10636 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1871234 0.89 ADORA1 (0.47) ADORA1ADORA3DRD2ADORA2B
SCHEMBL1875007 0.89 ADORA1 (0.55) ADORA1ADORA3DRD2ADORA2B
SCHEMBL1865267 0.87 ADORA1 (0.44) ADORA1ADORA3DRD2ADORA2B
SCHEMBL1866939 0.84 ADORA1 (0.44) ADORA1ADORA3ADORA2B
SCHEMBL1864689 0.83 ADORA1 (0.44) ADORA1ADORA3ADORA2BMAPT
SCHEMBL1870359 0.83 ADORA1 (0.44) ADORA1ADORA3ADORA2B
SCHEMBL1871730 0.83 ADORA1 (0.40) ADORA1ADORA3DRD2ADORA2B
SCHEMBL1861450 0.82 ADORA1 (0.49) ADORA1ADORA3ADORA2B
SCHEMBL1870705 0.82 ADORA1 (0.42) ADORA1ADORA3ADORA2B
SCHEMBL1866236 0.79 ADORA1 (0.41) ADORA1ADORA3ADORA2BMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2499142-A1 SUBSTITUTED FUSED PYRIMIDINE COMPOUNDS, ITS PREPARATION AND USES THEREOF Advinus Therapeutics Limited (IN) 2012-09-19 EP disclosed
WO-2011055391-A1 SUBSTITUTED FUSED PYRIMIDINE COMPOUNDS, ITS PREPARATION AND USES THEREOF ADVINUS THERAPEUTICS PRIVATE LIMITED (IN) 2011-05-12 WO disclosed