SCHEMBL1870359

SCHEMBL1870359

CCCn1c(Oc2cccc(CCO)c2)nc(=O)c2c1N=C(C1CCCC1)[N]2

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 13/20 0.44
ADORA3 P0DMS8 1/20 0.44
ADORA2B P29275 2/20 0.36
HSD11B1 P28845 1/20 0.35
ALPL P05186 1/20 0.34
KCNH2 Q12809 1/20 0.33
TRPC4 Q9UBN4 1/20 0.33
TRPC5 Q9UL62 1/20 0.33
ADORA2A P29274 1/20 0.33
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1875007 0.87 ADORA1 (0.55) ADORA1ADORA3ADORA2BALPLADORA2A
SCHEMBL1871234 0.84 ADORA1 (0.47) ADORA1ADORA3ADORA2BTRPC4TRPC5
SCHEMBL1864689 0.81 ADORA1 (0.44) ADORA1ADORA3ADORA2BADORA2A
SCHEMBL1870705 0.81 ADORA1 (0.42) ADORA1ADORA3ADORA2BADORA2A
SCHEMBL1861450 0.81 ADORA1 (0.49) ADORA1ADORA3ADORA2BADORA2AHCRTR2
SCHEMBL1869240 0.79 ADORA1 (0.38) ADORA1ADORA3ADORA2BADORA2A
SCHEMBL1869009 0.79 ADORA1 (0.47) ADORA1ADORA3ADORA2BALPL
SCHEMBL1871420 0.78 ADORA1 (0.41) ADORA1ADORA3ADORA2BADORA2A
SCHEMBL1866382 0.77 ADORA1 (0.57) ADORA1ADORA3ADORA2BADORA2A
SCHEMBL1865763 0.77 ADORA1 (0.37) ADORA1ADORA3ADORA2BADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2499142-A1 SUBSTITUTED FUSED PYRIMIDINE COMPOUNDS, ITS PREPARATION AND USES THEREOF Advinus Therapeutics Limited (IN) 2012-09-19 EP claimed
WO-2011055391-A1 SUBSTITUTED FUSED PYRIMIDINE COMPOUNDS, ITS PREPARATION AND USES THEREOF ADVINUS THERAPEUTICS PRIVATE LIMITED (IN) 2011-05-12 WO claimed
EP-2499142-A1 SUBSTITUTED FUSED PYRIMIDINE COMPOUNDS, ITS PREPARATION AND USES THEREOF Advinus Therapeutics Limited (IN) 2012-09-19 EP disclosed
WO-2011055391-A1 SUBSTITUTED FUSED PYRIMIDINE COMPOUNDS, ITS PREPARATION AND USES THEREOF ADVINUS THERAPEUTICS PRIVATE LIMITED (IN) 2011-05-12 WO disclosed