SCHEMBL18696182

SCHEMBL18696182

OCCN1C=C2C(Nc3ccc(OC(F)(F)F)cc3)NCNC2N1

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 7/20 0.35
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
ATM Q13315 1/20 0.35
ABL1 P00519 2/20 0.34
BCR P11274 2/20 0.34
ALDH1A1 P00352 2/20 0.34
LMNA P02545 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CHRNA7 P36544 1/20 0.34
ACHE P22303 1/20 0.33
GAA P10253 1/20 0.33
MAPK1 P28482 1/20 0.33
KDM4E B2RXH2 1/20 0.33
POLB P06746 1/20 0.33
MAPT P10636 1/20 0.33
EPHX1 P07099 1/20 0.32
P2RX3 P56373 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16374017 0.62 ABL1 (0.46) EPHX2KMT2AMEN1ATMABL1
SCHEMBL2172826 0.59 EPHX2 (0.51) EPHX2KDM4EMAPTEPHX1
SCHEMBL6289309 0.59 MAPT (0.55) EPHX2KMT2AMEN1ALDH1A1LMNA
SCHEMBL14916657 0.57 EPHX2 (0.56) EPHX2ALDH1A1KDM4EPOLBMAPT
SCHEMBL5536264 0.57 EPHX1 (0.64) EPHX2KMT2AMEN1ABL1BCR
Hydrochloric Acid SCHEMBL31155662 0.57 EPHX1 (0.47) EPHX2KMT2AMEN1ATMMAPT
SCHEMBL27912284 0.57 MAPT (0.59) EPHX2KMT2AMEN1ALDH1A1LMNA
Hydrochloric Acid SCHEMBL411544 0.56 EPHX1 (0.63) EPHX2KMT2AMEN1ALDH1A1MAPK1
SCHEMBL12175682 0.56 CARM1 (0.51) EPHX2ALDH1A1
SCHEMBL27268412 0.55 MAPT (0.57) EPHX2KMT2AMEN1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3150593-A1 SMALL MOLECULE MYRISTATE INHIBITORS OF BCR-ABL AND METHODS OF USE Dana Farber Cancer Institute, Inc. (US) 2017-04-05 EP disclosed