SCHEMBL18698252

SCHEMBL18698252

CCC(=O)c1cc(-c2cccc(Cl)c2)n[nH]1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALPL P05186 4/20 0.50
KDM5B Q9UGL1 1/20 0.49
MAPT P10636 5/20 0.49
GAA P10253 2/20 0.49
CA12 O43570 2/20 0.48
TP53 P04637 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.47
CHEK1 O14757 1/20 0.47
RET P07949 1/20 0.47
PDGFRB P09619 1/20 0.47
PIM1 P11309 1/20 0.47
PDGFRA P16234 1/20 0.47
GSK3B P49841 1/20 0.47
RPS6KA3 P51812 1/20 0.47
LIMK1 P53667 1/20 0.47
CDK5 Q00535 1/20 0.47
TYRO3 Q06418 1/20 0.47
MAPK14 Q16539 1/20 0.47
LRRK2 Q5S007 1/20 0.47
AURKB Q96GD4 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15933264 0.84 TP53 (0.51) ALPLKDM5BMAPTGAACA12
SCHEMBL25139711 0.84 TP53 (0.68) ALPLMAPTGAACA12TP53
SCHEMBL30716607 0.83 ALPL (0.74) ALPLMAPTGAATP53SMN1; SMN2
SCHEMBL16699171 0.83 ALPL (0.74) ALPLMAPTGAATP53SMN1; SMN2
SCHEMBL643921 0.82 TP53 (0.71) ALPLCA12TP53SMN1; SMN2CA9
SCHEMBL15930144 0.82 ADORA3 (0.51) ALPLKDM5BMAPTGAACA12
SCHEMBL18726283 0.81 SCN9A (0.54) ALPLKDM5BMAPTGAACA12
SCHEMBL644902 0.81 MAPT (0.72) ALPLMAPTGAASMN1; SMN2PLK1
SCHEMBL18648619 0.79 ALPL (0.58) ALPLMAPTGAASMN1; SMN2
SCHEMBL16711444 0.77 MAPT (0.53) ALPLKDM5BMAPTGAACA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9611274-B2 Macrocycles as factor XIa inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2017-04-04 US disclosed