SCHEMBL18699342

SCHEMBL18699342

O=Nc1ccc(/C=C/C(=O)/C(C(=O)/C=C/c2ccc(O)cc2)=C(O)/C=C/c2ccc(O)cc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYR P14679 3/20 0.50
CA2 P00918 3/20 0.50
AKR1B10 O60218 2/20 0.50
AKR1B1 P15121 2/20 0.50
PKM P14618 2/20 0.50
CA12 O43570 2/20 0.50
CA1 P00915 2/20 0.50
CA7 P43166 2/20 0.50
CA9 Q16790 2/20 0.50
CA14 Q9ULX7 2/20 0.50
ESR1 P03372 1/20 0.50
CA3 P07451 1/20 0.50
CA4 P22748 1/20 0.50
CA6 P23280 1/20 0.50
DPP4 P27487 1/20 0.50
CA5A P35218 1/20 0.50
HCAR2 Q8TDS4 1/20 0.50
ESR2 Q92731 1/20 0.50
CA5B Q9Y2D0 1/20 0.50
F3 P13726 3/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9974131 0.89 TYR (0.62) TYRCA2AKR1B10AKR1B1PKM
SCHEMBL15298982 0.78 CA12 (0.49) TYRCA2AKR1B10AKR1B1PKM
SCHEMBL25198993 0.76 F3 (0.77) PKMESR1ESR2F3TLR9
SCHEMBL25208467 0.76 F3 (0.77) PKMESR1ESR2F3TLR9
SCHEMBL16088502 0.72 MMP1 (0.62) TYRCA2AKR1B10AKR1B1PKM
SCHEMBL9972287 0.70 THRB (0.67) F3GSK3BBACE1MAOBCYP3A4
SCHEMBL107699 0.70
SCHEMBL19415817 0.70 GLA (0.59) TYRCA2AKR1B10AKR1B1PKM
SCHEMBL15483131 0.70 HDAC1 (0.54) TYRCA2AKR1B10AKR1B1PKM
Coumaric Acid SCHEMBL28320218 0.70 ESR1 (0.84) TYRCA2AKR1B10AKR1B1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3150203-B1 COMPOUNDS WITH (1E,6E)-1,7-BIS-(3,4- DIMETHOXYPHENYL)-4,4-DISSTITUTED-HEPA-1,6-DIENE-3,5-DI-ONE STRUCTURAL SCAFFOLD,THEIR BIOLOGICAL ACTIVITY, AND USES THEREOF ALLIANZ PHARMASCIENCE LTD (TW) 2020-02-19 EP disclosed
EP-3150203-A1 COMPOUNDS WITH (1E,6E)-1,7-BIS-(3,4- DIMETHOXYPHENYL)-4,4-DISSTITUTED-HEPA-1,6-DIENE-3,5-DI-ONE STRUCTURAL SCAFFOLD,THEIR BIOLOGICAL ACTIVITY, AND USES THEREOF Allianz Pharmascience Ltd (TW) 2017-04-05 EP disclosed