SCHEMBL18704182

SCHEMBL18704182

Cc1cc(N(C)C)nc(N)c1C#N

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.62
ALDH1A1 P00352 7/20 0.41
HPGD P15428 4/20 0.41
HSD17B10 Q99714 2/20 0.41
GAA P10253 1/20 0.41
PPARG P37231 1/20 0.39
STAT3 P40763 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
NR2E3 Q9Y5X4 1/20 0.39
NCOR2 Q9Y618 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
HTT P42858 3/20 0.38
TSHR P16473 1/20 0.38
RECQL P46063 1/20 0.38
IKBKB O14920 1/20 0.37
ADORA2A P29274 3/20 0.37
ADRA2A P08913 1/20 0.37
ADORA1 P30542 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8889388 0.79 L3MBTL1 (0.51) KDM4EALDH1A1HSD17B10GAANPSR1
SCHEMBL30411552 0.77 KDM4E (0.71) KDM4EALDH1A1HPGDHSD17B10GAA
SCHEMBL1140140 0.77 KDM4E (0.71) KDM4EALDH1A1HPGDHSD17B10GAA
SCHEMBL317616 0.77 KDM4E (1.00) KDM4EALDH1A1HPGDHSD17B10GAA
SCHEMBL25339386 0.74 KDM4E (0.67) KDM4EALDH1A1HPGDHSD17B10GAA
SCHEMBL11845115 0.74 KDM4E (0.67) KDM4EALDH1A1HPGDHSD17B10GAA
SCHEMBL29985618 0.74 KDM4E (0.67) KDM4EALDH1A1HPGDHSD17B10GAA
SCHEMBL18704154 0.71 KDM4E (0.49) KDM4EALDH1A1HPGDHSD17B10GAA
SCHEMBL17164131 0.71 RECQL (0.67) KDM4EALDH1A1HPGDHSD17B10GAA
SCHEMBL28806889 0.68 ADORA1 (0.71) KDM4EALDH1A1HPGDHSD17B10GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017060488-A1 NEW TRPA1 ANTAGONISTS ALMIRALL, S.A. (ES) 2017-04-13 WO disclosed