SCHEMBL1865267

SCHEMBL1865267

CCCn1c(OCc2cccc(C(F)(F)F)c2)nc(=O)c2c1N=C(C1CCCCC1)[N]2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 6/20 0.44
MAOB P27338 3/20 0.42
MAOA P21397 1/20 0.42
DRD2 P14416 1/20 0.37
HTR6 P50406 1/20 0.37
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
ALOX5AP P20292 1/20 0.36
FEN1 P39748 1/20 0.36
HCAR2 Q8TDS4 1/20 0.36
DRD4 P21917 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
ADORA2B P29275 2/20 0.35
ALDH1A1 P00352 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CARM1 Q86X55 1/20 0.35
PRMT6 Q96LA8 1/20 0.35
HSD11B1 P28845 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
ADORA2A P29274 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1870513 0.87 ADORA1 (0.58) ADORA1DRD2ADORA2BADORA3
SCHEMBL1871730 0.79 ADORA1 (0.40) ADORA1DRD2ALOX5APFEN1DRD4
SCHEMBL1871234 0.78 ADORA1 (0.47) ADORA1DRD2DRD4ADORA2BADORA3
SCHEMBL1875007 0.77 ADORA1 (0.55) ADORA1DRD2ADORA2BADORA3ADORA2A
SCHEMBL1866092 0.77 PDE5A (0.33) MAOBMAOAALOX5APFEN1SIGMAR1
SCHEMBL1866939 0.77 ADORA1 (0.44) ADORA1ADORA2BHSD11B1ADORA3ADORA2A
SCHEMBL1870359 0.76 ADORA1 (0.44) ADORA1ADORA2BHSD11B1ADORA3ADORA2A
SCHEMBL1871420 0.76 ADORA1 (0.41) ADORA1ADORA2BADORA3ADORA2A
SCHEMBL1868348 0.76 ADORA1 (0.58) ADORA1ADORA2BADORA2A
SCHEMBL1866236 0.75 ADORA1 (0.41) ADORA1ADORA2BALDH1A1ADORA3ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2499142-A1 SUBSTITUTED FUSED PYRIMIDINE COMPOUNDS, ITS PREPARATION AND USES THEREOF Advinus Therapeutics Limited (IN) 2012-09-19 EP claimed
WO-2011055391-A1 SUBSTITUTED FUSED PYRIMIDINE COMPOUNDS, ITS PREPARATION AND USES THEREOF ADVINUS THERAPEUTICS PRIVATE LIMITED (IN) 2011-05-12 WO claimed